Onconova Therapeutics, Inc. to Present New Data on Briciclib and Next-Generation CDK4/6 Inhibitor, ON 123300, at 2015 AACR-NCI-EORTC Meeting

On October 29, 2015 Onconova Therapeutics, Inc. (NASDAQ:ONTX), a clinical-stage biopharmaceutical company focused on discovering and developing novel products to treat cancer, reported the presentation of new non-clinical data for two of the Company’s proprietary compounds at the 2015 AACR (Free AACR Whitepaper)-NCI-EORTC AACR-NCI-EORTC (Free AACR-NCI-EORTC Whitepaper) International Conference on Molecular Targets and Cancer Therapeutics (EORTC-NCI-AACR) (Free ASGCT Whitepaper) (Free EORTC-NCI-AACR Whitepaper), which will be held November 5-9, 2015, in Boston, MA (Press release, Onconova, OCT 29, 2015, View Source [SID:1234507843]).

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A poster relating to the novel eIF4E targeted mechanism of action for briciclib, currently in a dose-escalating Phase 1 clinical trial in patients with advanced solid tumors refractory to current therapies, will be presented by Onconova’s collaborators from Harvard University. Another poster will highlight the developmental studies aimed at advancing the Company’s novel CDK4/6 inhibitor, ON 123300, towards an Investigational New Drug (IND) Application filing. The presentations are listed below.

Mechanism of action studies for briciclib

Abstract number: B126
Title: Targeted inhibition of eIF4E-mediated translation by the novel small molecule anti-cancer compound, briciclib (ON 013105).
Date: Saturday, 11/7/2015
Time: 12:30 PM — 3:30 PM ET
Location: Session B, Hall C-D

IND-directed studies for next-generation CDK4/6 inhibitor ON 123300

Abstract number: LB-A21
Title: Single-agent activity and favorable pharmaceutical properties of orally bioavailable next-generation CDK4/6 inhibitor, ON 123300.
Date: Friday, 11/6/2015
Time: 12:15 PM — 3:15 PM ET
Location: Session A, Hall C-D

Seattle Genetics Reports Third Quarter 2015 Financial Results

On October 29, 2015 Seattle Genetics, Inc. (Nasdaq: SGEN) reported financial results for the third quarter and nine months ended September 30, 2015 (Press release, Seattle Genetics, OCT 29, 2015, View Source;p=RssLanding&cat=news&id=2104338 [SID:1234507844]). The company also highlighted ADCETRIS (brentuximab vedotin) commercialization, regulatory and clinical development accomplishments, progress with other proprietary pipeline programs and antibody-drug conjugate (ADC) collaborator updates.

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"We are pleased to have delivered on several key milestones recently, including an expanded label for ADCETRIS based on our phase 3 AETHERA trial, completing enrollment in the ALCANZA phase 3 trial and reaching our target enrollment in the phase 3 ECHELON-1 trial," said Clay Siegall, Ph.D., President and Chief Executive Officer of Seattle Genetics. "We also completed a successful public offering in September that strongly positions us to continue investing in expanding the ADCETRIS opportunity, advancing our product pipeline and conducting innovative research. We are preparing for a strong presence at the upcoming ASH (Free ASH Whitepaper) annual meeting with data from ADCETRIS, SGN-CD33A and other pipeline programs."

Recent ADCETRIS Highlights

Received regular approval from the U.S. Food and Drug Administration (FDA) for ADCETRIS (brentuximab vedotin) for classical Hodgkin lymphoma (HL) patients at high risk of relapse or progression as post-autologous transplant consolidation based on the phase 3 AETHERA clinical trial. The approval represents the third indication for ADCETRIS in the United States. The AETHERA trial also converted the prior accelerated approval of ADCETRIS in relapsed HL to regular approval.

Completed enrollment in the phase 3 ALCANZA clinical trial for patients with CD30-expressing cutaneous T-cell lymphoma (CTCL) who have received prior systemic therapy. The randomized trial is evaluating ADCETRIS versus investigator’s choice of methotrexate or bexarotene in 132 patients. Data are anticipated in the second half of 2016.

Completed target patient enrollment in the phase 3 ECHELON-1 clinical trial. ECHELON-1 is a randomized trial evaluating ADCETRIS as part of a frontline combination chemotherapy regimen in patients with previously untreated advanced classical HL.
Initiated a randomized phase 2 trial of rituximab (Rituxan) and bendamustine (Treanda) with or without ADCETRIS for relapsed or refractory patients with CD30-expressing diffuse large B-cell lymphoma (DLBCL).

Initiated a phase 1/2 clinical trial of ADCETRIS in combination with nivolumab (Opdivo) for patients with relapsed or refractory HL after failure of frontline treatment. The trial is being conducted under a previously announced clinical trial collaboration agreement with Bristol-Myers Squibb Company.

Recent Pipeline, Collaborator and Other Highlights

Initiated a randomized phase 2 trial of SGN-CD19A (denintuzumab mafodotin) in combination with the second-line salvage regimen of rituximab, ifosfamide, carboplatin and etoposide (RICE) for patients with relapsed or refractory DLBCL.

Submitted an investigational new drug (IND) application to the FDA for SGN-CD19B, a CD19-targeted ADC utilizing the company’s pyrrolobenzodiazepine (PBD) dimer cell-killing agent and proprietary site-specific conjugation technology (EC-mAb). A phase 1 trial is planned in the first half of 2016.

Expanded our 2011 collaboration with AbbVie to provide access to Seattle Genetics’ PBD dimer and EC-mAb technology. Financial terms were not disclosed.

Received a milestone payment under our collaboration with AbbVie, triggered by its initiation of a phase 1 trial for an auristatin-based ADC for solid tumors utilizing Seattle Genetics’ technology.

Added to and promoted several members of the senior management team, including:
Promoting Elaine Waller, PharmD, to Executive Vice President, Regulatory Affairs and Clinical Development Operations. Dr. Waller has been with Seattle Genetics since September 2008. She has led numerous successful regulatory initiatives for the company, including the recent ADCETRIS label expansion.

Promoting Peter Senter, Ph.D., to Vice President, Chemistry and Senior Distinguished Fellow. Dr. Senter joined Seattle Genetics in August 1998. As an early member of the company’s research organization, he has contributed significantly to Seattle Genetics’ leadership position in ADCs and the innovative science behind its pipeline programs.

Hiring Rachel Lenington as Vice President, Program, Portfolio and Alliance Management. Ms. Lenington previously spent five years at the Bill & Melinda Gates Foundation focused on global health strategies, product development and alliances. Before that she spent 10 years at Amgen.

Hiring Matt Skelton as Vice President, Marketing. Mr. Skelton previously spent 16 years at Amgen in a range of sales and marketing roles. Before that, he was at Eli Lilly.

Promoting Phil Tsai, Ph.D., to Vice President, Process Sciences. Dr. Tsai has been at Seattle Genetics since January 2003. During his tenure, he has led the development of many antibody and ADC manufacturing processes at various stages of the product development life cycle.

Anticipated Upcoming Activities

ADCETRIS

Report ADCETRIS data from multiple clinical trials at the American Society of Hematology (ASH) (Free ASH Whitepaper) 2015 Annual Meeting, being held December 5-8, 2015 in Orlando, FL:
ADCETRIS in HL, including five-year survival data from a pivotal trial in relapsed/refractory patients, data from phase 2 trials in the second-line salvage setting and in the frontline setting for patients age 60 or older, and updated efficacy and safety data from the AETHERA phase 3 trial;
ADCETRIS in non-Hodgkin lymphoma, including frontline and relapsed DLBCL and long-term follow up from a phase 1 trial of ADCETRIS in combination with chemotherapy in T-cell lymphomas; and,
Data from numerous investigator-sponsored trials of ADCETRIS in various lymphoma settings and combinations.
Initiate a phase 1/2 trial of ADCETRIS in combination with nivolumab for relapsed non-Hodgkin lymphoma.
Complete enrollment in phase 3 ECHELON-2 trial during 2016.

ADCETRIS is not currently approved for use in frontline HL, second-line HL, CTCL, DLBCL or non-Hodgkin lymphoma other than systemic anaplastic large cell lymphoma.

SGN-CD33A (Vadastuximab Talirine)

Receive feedback from the FDA and European regulators regarding our regulatory strategy for SGN-CD33A in acute myeloid leukemia (AML).

Report data at ASH (Free ASH Whitepaper) from phase 1 trials of SGN-CD33A in AML, including as monotherapy and in combination with hypomethylating agents (HMAs).

Initiate a phase 1/2 trial of SGN-CD33A as pre-conditioning or post-allogeneic transplant maintenance treatment in patients with AML in the first half of 2016.

Initiate a phase 1/2 trial with SGN-CD33A in combination with azacitidine (Vidaza) for patients with previously untreated myelodysplastic syndrome (MDS) in the first half of 2016.

Other Pipeline Programs

Report data from pipeline programs at ASH (Free ASH Whitepaper):
Phase 1 trials of SGN-CD19A in non-Hodgkin lymphoma and acute leukemia; and,
Preclinical studies of two novel ADCs, SGN-CD19B and SGN-CD123A, which are expected to advance into clinical trials in 2016 for non-Hodgkin lymphoma and AML, respectively.

Report interim phase 1 clinical data from SGN-LIV1A, an ADC targeted to LIV-1 in development for metastatic breast cancer, at the San Antonio Breast Cancer Symposium being held December 8-12, 2015 in San Antonio, TX.

Initiate a randomized phase 2 trial of SGN-CD19A in frontline DLBCL in the first half of 2016.

Report phase 1 clinical data from ASG-15ME and ASG-22ME (enfortumab vedotin) in the first half of 2016. These programs are in development for solid tumors, notably bladder cancer, under a collaboration with Astellas.

Initiate a phase 1 trial of SGN-CD19B in non-Hodgkin lymphoma in the first half of 2016.

Third Quarter and Nine Months 2015 Financial Results

Total revenues in the third quarter and nine month periods ended September 30, 2015 increased to $84.1 million and $243.3 million, respectively, from $75.9 million and $212.4 million for the same periods in 2014. Revenues were derived from:

ADCETRIS sales in the third quarter of $59.1 million, an increase from $48.2 million in the third quarter of 2014. For the year-to-date, ADCETRIS sales were $163.0 million, compared to $131.7 million for the year-to-date period in 2014, a 24 percent increase.
Royalty revenues in the third quarter of 2015 were $9.7 million, compared to $8.1 million in the third quarter of 2014. For the year-to-date in 2015, royalty revenues were $28.4 million, compared to $28.2 million for the first nine months of 2014. Royalty revenues are primarily driven by international sales of ADCETRIS by Takeda. First quarter 2014 royalty revenues included a $5.0 million sales milestone payment from Takeda.

Amounts earned under the company’s ADCETRIS and ADC collaborations totaled $15.3 million in the third quarter and $51.9 million for the first nine months of 2015, compared to $19.5 million and $52.6 million for the same periods in 2014.
Total costs and expenses for the third quarter of 2015 were $110.6 million, compared to $91.5 million for the third quarter of 2014. For the first nine months of 2015, total costs and expenses were $339.1 million, compared to $262.1 million in the first nine months of 2014. The increase in 2015 costs and expenses was primarily driven by investment in Seattle Genetics’ pipeline programs, including a $25.0 million upfront payment made in the second quarter of 2015 as part of our collaboration with Unum Therapeutics.

Non-cash, share-based compensation cost for the first nine months of 2015 was $28.7 million, compared to $29.0 million for the first nine months of 2014.

Net loss for the third quarter of 2015 was $26.4 million, or $0.21 per share, compared to a net loss of $15.6 million, or $0.13 per share, for the third quarter of 2014. For the nine months ended September 30, 2015, net loss was $95.6 million, or $0.76 per share, compared to a net loss of $49.5 million, or $0.40 per share, for the same period in 2014.

As of September 30, 2015, Seattle Genetics had $736.5 million in cash, cash equivalents and investments, compared to $313.4 million as of December 31, 2014. The increase in cash and investments reflects net proceeds of approximately $526.6 million from the company’s public offering of common stock that closed on September 16, 2015.

2015 Financial Outlook

Seattle Genetics anticipates that 2015 revenues from ADCETRIS net product sales in the U.S. and Canada will be higher than previously anticipated, and are now expected to be in the range of $218 million to $223 million.

Third quarter results 2015

On October 29, 2015 Sanofi Chief Executive Officer, Olivier Brandicourt, reported:
"The Group showed growth on both top and bottom line in the third quarter driven by strong performance of Genzyme, Vaccines and Emerging Markets (Press release, Sanofi, OCT 29, 2015, View Source [SID:1234507915]). At the same time, we continue to make significant investments to strengthen Sanofi for the future. With the growing adoption of new products such as Aubagio, NexGard, Lemtrada, and Toujeo and the recent launch of Praluent, we have achieved important milestones in our mission to bring innovative medicines to patients. Despite headwinds in our diabetes business, we are confident in Sanofi’s long-term prospects and we look forward to sharing our roadmap for the Group on November 6, 2015."

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(1) In order to facilitate an understanding of operational performance, Sanofi comments on the business net income statement. Business net income is a non-GAAP financial measure (See Appendix 8 for definitions of financial indicators). The consolidated income statement for Q3 2015 is provided in Appendix 4 and a reconciliation of business net income to IFRS net income reported in Appendix 3; (2) Percentage changes in net sales are expressed at constant exchange rates (CER) unless otherwise indicated (see Appendix 8 for a definition); (3) See page 8; (4) 2014 business EPS was €5.20

2015 third-quarter and 9-month sales

Unless otherwise indicated, all percentage changes in sales in this press release are stated at constant exchange rates(1).

Third quarter sales of Sanofi increased 9.2% on a reported basis to €9,591 million. Exchange rate movements had a positive effect of 5.8 percentage points reflecting mainly the strength of the U.S. dollar and Chinese Yuan against the Euro which largely offset the Venezuelan Bolivar, the Brazilian real and Russian Ruble negative impact. At constant exchange rates, sales increased 3.4%.

Year-to-date sales were €27,779 million, an increase of 12.5% on a reported basis. Exchange rate movements had a favorable effect of 8.9 percentage points.

Pharmaceuticals

In the third quarter, sales for Pharmaceuticals increased 2.6% to €7,267 million, driven by Genzyme, which were partially offset by lower sales of Diabetes. Year-to-date sales for Pharmaceuticals were €22,522 million, up 2.8%.

In the third quarter, sales of the Diabetes division decreased 6.6% to €1,852 million, reflecting lower sales of Lantus in the U.S. In the U.S., sales of Diabetes were €1,075 million (down 16.4%). Sales of Diabetes outside the U.S. were €777 million, an increase of 8.1%. Strong performance in Emerging Markets (€373m, up 15.5%) was moderated by stable sales in Western Europe (€296m, down 0.3%), largely attributable to the entry of glargine biosimilar competition. Year-to-date sales for the Diabetes division were €5,677 million down 4.6%.

Given recent sales trends for the diabetes business and ongoing market dynamics, Sanofi now expects its global diabetes sales to be down between 6% to 7% at CER for 2015. Accounting for recent market trends, Sanofi now projects global diabetes sales over the period of 2015-2018 to decline at an average annualized rate of between 4% and 8% at CER. Approximately half of this revision is linked to insulin glargine and the other half is related to reduced expectations for Afrezza, Lyxumia and BGM (Blood Glucose Monitoring). Sanofi will mitigate the impact of this revised sales expectation on its business operating income by 2018 and will present the mid-term strategic and financial outlook for the Group on November 6, 2015.

Third-quarter sales of Lantus were €1,561 million down 10.8%. In the U.S., sales of Lantus decreased 19.6% to €997 million mainly due to a slowdown of basal insulin market growth, continued higher discounts on Lantus as compared to last year and unfavorable mix effect towards government channels such as Medicaid. In Western Europe, sales of the product decreased 1.4% to €222 million over the period. A biosimilar of Lantus from Eli Lilly was launched in several European markets in the third quarter (including Germany, UK, Netherlands, and Denmark) and in Japan. In Emerging Markets, third-quarter sales of Lantus were up 15.8% to €260 million, driven by China. Year-to-date sales of Lantus decreased 7.3% to €4,854 million.

In September, Sanofi reached a settlement agreement with Eli Lilly. The agreement resolves a U.S. patent infringement lawsuit regarding Lilly’s pursuit of regulatory approval for a product that would compete with Lantus SoloSTAR. Sanofi and Lilly agreed to end that lawsuit and to discontinue similar disputes worldwide. Under the agreement, Lilly will pay royalties to Sanofi in exchange for a license to certain Sanofi patents. In the U.S., Lilly will not sell its insulin glargine product before December 15, 2016.

Toujeo, a next-generation basal insulin, was launched in the U.S. market at the end of March and has rapidly obtained market access comparable to Lantus. After the first full two quarters on the market, Toujeo performance is encouraging. The product is trending favorably compared to diabetes analogue launches and now captures around 14% of IMS basal market NBRx share (New-to-Brand Prescriptions) in the U.S. Following EMA approval in April, Toujeo was recently launched in Germany, the U.K., the Netherlands and several Nordic countries where the uptake of the product has shown early promise. Toujeo was also recently launched in Japan and Canada. Total sales of the product were €46 million in the third quarter compared to €13 million in the second quarter of 2015. In the first nine months of 2015, sales of Toujeo were €66 million.

In the third quarter, sales of Amaryl increased 5.7% to €93 million, of which €75 million were generated in Emerging Markets (up 13.6%). Year-to-date sales of Amaryl were up 2.2% to €299 million. Third-quarter sales of Apidra were €88 million, down 4.5%, reflecting lower sales in the U.S. (-17.1% to €34 million). In Emerging Markets, sales of Apidra increased 16.7% to €19 million.
Year-to-date sales of Apidra were up 5.4% to €272 million. Afrezza sales were €2 million and €5 million in the third quarter and the first nine months of 2015, respectively.

Praluent

In September, the European Commission granted marketing authorization for Praluent (alirocumab, collaboration with Regeneron) for the treatment in certain adult patients of hypercholesterolemia characterized by high level of low-density lipoprotein (LDL) cholesterol. This approval follows the FDA approval received on July 24th, 2015. Praluent was launched in July in the U.S. and, as the product gains market access and awareness develops within the broader medical community, the uptake is expected to be gradual. Initial market access success includes the decision by Express Scripts to add Praluent in a branded preferred Tier 2 formulary position. Sales of Praluent were €4 million in Q3 2015.

Genzyme

Third-quarter sales of Genzyme grew 32.7% to €923 million boosted by the strong performance of Aubagio and the launch progress of Lemtrada. Genzyme recorded another quarter with double-digit sales growth in all territories; U.S. sales increased 40.2% to €431 million, Western Europe sales grew 29.5% to €271 million and Emerging Markets sales were up 27.7% to €135 million. Year-to-date sales of Genzyme increased 30.0% to €2,651 million.

Sales of Rare Diseases were up 13.0% to €630 million in the third-quarter.

Sales of the Gaucher franchise grew 14.3% to €207 million in the third-quarter. In the U.S. sales of this franchise were up 25.0% to €71 million. Sales of Cerezyme were €189 million up 5.1% sustained by Emerging Markets (up 20.0% to €62 million). In the U.S., sales of Cerezyme were down 4.2% reflecting the launch of Cerdelga, the only first-line oral therapy for Gaucher disease type 1 patients. Sales of Cerdelga reached €18 million in the third quarter of which U.S. sales accounted for €16 million. Year-to-date sales of Cerezyme increased 5.4% to €577 million and year-to-date sales of Cerdelga were €44 million.

Third-quarter sales of Fabrazyme grew 18.1% to €147 million. The product recorded strong performance in all territories reflecting new patients accrual; U.S. sales were up 12.1% to €76 million, Western Europe sales grew 21.4% to €34 million, Emerging Markets sales increased 30.8% to €15 million and the Rest of the World sales were up 23.5% to €22 million. Year-to-date sales of Fabrazyme increased 16.0% to €434 million.

Third-quarter sales of Myozyme/Lumizyme were up 10.9% to €162 million driven by the U.S. (up 25.7% to €51 million) which was sustained by the continued accrual of new patients. In Emerging Markets, sales increased 8.7% to €25 million and in Western Europe sales were up 7.2% to €75 million. Year-to-date sales of Myozyme/Lumizyme were €483 million, an increase of 14.5%.

Sales of Multiple Sclerosis products increased 120.2% to €293 million in the third quarter.

Third-quarter sales of Aubagio grew 78.6% to €225 million driven by sales in the U.S. (up 54.0% to €159 million) and Western Europe (€52 million versus €18 million in the same period of 2014) sustained by strong performance in France. Magnetic resonance imaging data from TEMSO study presented at ECTRIMS in October, demonstrate that Aubagio significantly slowed the brain volume loss (or atrophy) vs. placebo over two years in people with relapsing multiple sclerosis. Year-to-date sales of Aubagio increased 81.9% to €599 million.

Sales of Lemtrada were €68 million in the third quarter including €39 million in the U.S. and €22 million in Western Europe (mainly in Germany and the UK). Investigational data from the extension study presented at ECTRIMS support the value proposition of Lemtrada showing that the treatment effects were maintained over five years in the majority of patients with Relapsing Remitting Multiple Sclerosis. Year-to-date sales of Lemtrada were €162 million compared to €18 million in the first nine months of 2014.

Consumer Healthcare

Third-quarter sales of Consumer Healthcare (CHC) products were €814 million, an increase of 3.2% driven by Allegra, Lactacyd, and Dorflex. Sales of CHC in the U.S. grew 10.8% to €209 million. Sales of CHC in Emerging Markets were up 2.0% to €393 million driven by a low basis for comparison in Brazil and partially offset by lower sales in China. In Western Europe, sales decreased 7.6% to €146 million impacted by lower sales of Doliprane in France where price decreased in January 2015. In the Rest of the World, sales grew 20.7% to €66 million, reflecting good performance in Australia. Year-to-date sales of CHC reached €2,683 million, an increase of 3.3%.

Generics

Sales of Generics increased 6.7% to €452 million in the third quarter driven by sales of the authorized generics of Lovenox in the U.S. as well as Plavix in Japan which was launched by Sanofi and its partner Nichi-Iko Pharmaceuticals at the end of Q2 2015. In Emerging Markets and Western Europe sales of Generics increased 4.5% (to €262 million) and 5.6% (to €135 million), respectively. Year-to-date sales of Generics increased 8.7% to €1,450 million.

Oncology

Third-quarter sales of Oncology were up 5.4% to €376 million driven by Eloxatin in China and the U.S., Jevtana in the U.S. and Japan. Year-to-date sales of Oncology were €1,123 million, up 0.5%.

Sales of Jevtana increased 9.0% to €78 million in the third quarter led by the U.S. (up 13% to €32 million) and Japan where the product was launched in September 2014. Year-to-date sales of Jevtana were up 10.1% to €237 million.

Sales of Thymoglobulin increased 5.6% to €63 million and 3.8% to €187 million in the third quarter and the first nine months of 2015, respectively.

Third-quarter sales of Eloxatin were up 27.9% (to €58 million) sustained by growth in China and the U.S. Over the same period, sales of Taxotere decreased 3.4% (to €58 million), mainly due to generic competition in Japan. Year-to-date sales of Eloxatin and Taxotere were up 12.5% (€169 million) and down 17.9% (€173 million), respectively.

Sales of Mozobil grew 13.8% (to €36 million) and 17.5% (to €105 million) in the third quarter and the first nine months of 2015, respectively.

Established Rx Products

Total sales of Established Rx Products were stable (up 0.1%) at €2,846 million in the third quarter.

Sales of Plavix decreased 5.3% to €446 million in the third quarter reflecting generic competition in Japan in June 2015 (sales in Japan were down 24.7% to €145 million) partially offset by strong performance in China (up 17.6%) and Middle-East. Year-to-date sales of Plavix decreased 0.4% to €1,474 million.

Third-quarter sales of Lovenox were €429 million, up 0.9%. The product recorded a strong performance in Emerging Markets (up 17.0% to €167 million) driven by Africa, Middle-East and Brazil which offset the impact of generic competition in the U.S. (down 61.8% to €16 million). In Western Europe, sales were down 0.9% to €221 million. Sanofi is aware of competitors that have filed marketing authorization applications for biosimilar enoxaparin with health authorities in Europe. Year-to-date sales of Lovenox were €1,300 million (up 0.6%).

Sales of Renvela/Renagel increased 27.8% to €239 million in the third-quarter driven by growth in the U.S. (up 56.3% to 191 million) which benefited from a low third quarter 2014 comparison due to a limited allotment of generic Renvela tablets granted to Impax. Sales of Renvela/Renagel were down 28.6% to €15 million in Emerging Markets and down 18.8% to €26 million in Western Europe. Generics are currently marketed in some European countries and Sanofi continues to expect potential generic approvals in the U.S. Year-to-date sales of Renvela/Renagel grew 27.0% to €696 million.

Sales of Aprovel/Avapro decreased 8.4% to €167 million in the third quarter reflecting generic competition in Western Europe (down 22.0% to €32 million). In Emerging Markets, sales of the product were down 3.0% to €97 million. The performance in China was partially offset by Latin America. Year-to-date sales of Aprovel/Avapro were €592 million (down 2.4%).

Vaccines

Consolidated sales of Sanofi Pasteur increased 5.5% to €1,717 million in the third quarter driven by Polio/Pertussis/Hib vaccines in Emerging Markets, Menactra in the U.S. and VaxServe (a Sanofi Pasteur company and U.S. specialty supplier of vaccines). Third-quarter sales of Sanofi Pasteur increased 6.5% (to €1,198 million) in the U.S. and 22.3% (to €358 million) in Emerging Markets. Year-to-date sales of Sanofi Pasteur increased 4.0% to €3,301 million.

Third-quarter sales of Influenza vaccines increased 0.3% to €736 million. The performance in the U.S. (up 8.3% to €576 million) reflects Sanofi Pasteur’s strategy to offer a range of differentiated influenza vaccines. Sales in Emerging Markets were down 23.9% to €71 million as a result of delayed supply in Mexico. Western Europe sales were down 18% to €73 million. Year-to-date sales of Influenza vaccines decreased 7.1% to €872 million reflecting lower sales in Brazil due to increased supply of the Butantan Institute as a result of the technology transfer agreement with Sanofi Pasteur.

Third-quarter sales of Polio/Pertussis/Hib vaccines were up 17.8% to €327 million driven by Pentaxim, the ramp up of Hexaxim and polio vaccines. In Emerging Markets, sales of Polio/Pertussis/Hib vaccines increased 62.4% to €195 million boosted by sales of Pentaxim and Polio vaccines in China. In the U.S. sales of Polio/Pertussis/Hib vaccines decreased 13.4% to €100 million due to lower sales of Pentacel. Over the period, Shantha sold €5 million of Shan5TM, its pediatric pentavalent vaccine, to global health organizations. Year-to-date sales of Polio/Pertussis/Hib vaccines increased 5.2% to €882 million.

Sales of Menactra grew 17.8% to €239 million in the third quarter reflecting higher U.S. public sector sales. Year-to-date sales of Menactra increased 18.7% to €459 million.

Third-quarter sales of Adult Booster vaccines were €133 million, down 9.9% and reflecting lower sales in Western Europe (down 53.6% to €13 million) due to phasing effect. Year-to-date sales of Adult Booster vaccines were €346 million, an increase of 1.4%.

Third-quarter and Year-to-date sales of Travel and Other Endemic Vaccines declined 8.1% to €96 million and 8.7% to €275 million, respectively.

Sales of Sanofi Pasteur MSD (not consolidated), the joint venture with Merck & Co. in Europe, were €284 million (down 3.7% on a reported basis) and €584 million (down 3.9% on a reported basis) in the third quarter and first nine months, respectively.

Animal Health

Third-quarter sales of Animal Health increased 9.3% to €607 million driven by the continued success of NexGard, Merial’s new generation flea and tick product for dogs and also supported by strong performance of our Avian franchise. In the U.S. and Emerging Markets, Animal Health sales grew 10.9% (to €289 million) and 14.0% (to €151 million), respectively. Year-to-date sales of Animal Health increased 12.4% to €1,956 million.

Sales of the Companion Animals segment were up 13.6% to €401 million in the third quarter, as a result of NexGard. The performance of NexGard more than offset the decline in sales of the Frontline products family. Year-to-date sales of Companion Animals segment grew 14.3% to €1,308 million.

Third-quarter sales of the Production Animals segment increased 2.5% to €206 million driven by the Avian business in Emerging Markets. Year-to-date sales of the Production Animals segment grew 8.9% to €648 million.

Net sales by geographic region

World less the U.S., Canada, Western Europe, Japan, South Korea, Australia and New Zealand;
France, Germany, UK, Italy, Spain, Greece, Cyprus, Malta, Belgium, Luxembourg, Portugal, Netherlands, Austria, Switzerland, Sweden, Ireland, Finland, Norway, Iceland, Denmark;
Japan, South Korea, Canada, Australia and New Zealand;
Sales in the U.S. increased 2.3% to €3,888 million in the third quarter. The performance of Genzyme (up 40.2%), Vaccines (up 6.5%), CHC (up 10.8%), Animal Health (up 10.9%), and Oncology (up 10.4%) was partially offset by lower sales of Diabetes (down 16.4%). Year-to-date sales in the U.S. grew 1.8% to €10,114 million.

Third-quarter sales in Emerging Markets grew 11.4% to 2,871 million due to the performance of Pharmaceuticals (up 9.9%), Vaccines (up 22.3%) and Animal Health (up 14.0%). In Pharmaceuticals, double-digit growth over the period was delivered by Diabetes (up 15.5%), Genzyme (up 27.7%) Oncology (up 13.8%) and Established Rx products (up 10.7%). In Asia, third-quarter sales were up 17.8% to €964 million, boosted by the performance in China (up 33.2% to €593 million). In China, the performance was largely attributable to Vaccines, Plavix, Lantus, Aprovel and Eloxatin. In Latin America, third-quarter sales were up 7.0% to €697 million. Third-quarter sales in Brazil increased 10.1% to €270 million. Sales in Eastern Europe, Russia and Turkey grew 6.0% to €587 million in the third quarter driven by Turkey and Ukraine. Sales in Russia were up 2.1% to €137 million, reflecting the local economic situation. In Africa and Middle-East, sales grew 11.4% to €562 million. In the Emerging Markets, year-to-date sales increased 8.7% to €8,912 million.

Sales in Western Europe were €1,988 million, down 1.8% in the third quarter. Strong performance of Genzyme (up 29.5%), was offset by lower sales of Established Rx products (-6.3%), CHC (-7.6%) and Vaccines (-24.1%). Year-to-date sales in Western Europe increased 0.6% to €6,017 million.

In the third quarter, sales in Japan decreased 11.4% to €458 million, reflecting generic competition to Plavix (-24.7%) and lower sales of Vaccines (-38.7%). In Japan, year-to-date sales decreased 4.0% to €1,572 million.

R&D update

Consult Appendix 6 for full overview of Sanofi’s R&D pipeline
Regulatory update

Regulatory updates since the publication of the second quarter results on July 30, 2015 include the following:

In October, VaxiGrip QIV (Quadrivalent inactivated influenza vaccine) for children three years old or above was submitted to European authorities.
In September, the U.S. Food and Drug Administration (FDA) accepted for filing the New Drug Application (NDA) for lixisenatide, an investigational once-daily prandial GLP-1 receptor agonist for the treatment of adults with type 2 diabetes.
In September, the European Commission (EC) granted marketing authorization for Praluent (alirocumab, collaboration with Regeneron) for the treatment in certain adult patients of hypercholesterolemia characterized by high level of low-density lipoprotein (LDL) cholesterol. This approval follows the FDA approval received on July 24th. In August, Praluent was also submitted to Japanese health authorities.
At the end of October 2015, the R&D pipeline contained 41 pharmaceutical new molecular entities (excluding Life Cycle Management) and vaccine candidates in clinical development of which 13 are in Phase III or have been submitted to the regulatory authorities for approval.

Collaboration

In August, Sanofi and Google Life Sciences announced that the companies are collaborating to improve care and outcomes for people with type 1 and type 2 diabetes. The collaboration will pair Sanofi’s leadership in diabetes treatments and devices with Google’s expertise in analytics, miniaturized electronics and low power chip design. The companies will explore how to improve diabetes care by developing new tools that bring together many of the previously siloed pieces of diabetes management and enable new kinds of interventions. This includes health indicators such as blood glucose and hemoglobin A1c levels, patient-reported information, medication regimens and sensor devices.
In August, Sanofi also entered a research collaboration and license agreement with Evotec and Apeiron Biologics to discover and develop first-in-class small molecule-based immuno-oncology therapies to treat solid and hematological cancers by enhancing the anti-tumor activity of the human immune system.
In August, Sanofi entered a strategic research collaboration with Evotec to develop beta cell-modulating diabetes treatments, which may reduce or eliminate the need for insulin injections.
Portfolio update

Phase III:

Positive new five-year investigational data from the extension study of Lemtrada (alemtuzumab) for patients with relapsing remitting multiple sclerosis were presented in October at ECTRIMS.

New analysis from the Phase III TEMSO study was presented on October at ECTRIMS. Magnetic resonance imaging (MRI) data from TEMSO demonstrate that Aubagio significantly slowed brain volume loss (or atrophy) vs. placebo over two years in people with relapsing multiple sclerosis. In this analysis, MRI data from TEMSO were analyzed utilizing SIENA (structural image evaluation using normalization of atrophy), an alternative methodology than the one originally used.

In September, Sanofi announced that the LixiLan-L Phase III clinical trial met its primary endpoint in patients with type 2 diabetes treated with insulin glargine with or without metformin. The fixed-ratio combination of insulin glargine 100 Units/mL and lixisenatide, a GLP-1 receptor agonist, demonstrated statistically superior reduction in HbA1c compared with insulin glargine 100 Units/mL. Overall, the fixed-ratio combination had a safety profile reflecting those of insulin glargine 100 Units/mL and lixisenatide. In July, Sanofi announced also that the first LixiLan Phase III study, LixiLan-O, met its primary objective in patients with type 2 diabetes treated with metformin. Regulatory submissions are planned for Q4 2015 in the United States and Q1 2016 in the European Union.

A new pooled analysis of heterozygous familial hypercholesterolemia (HeFH) patients included in the ODYSSEY clinical trial program showed that Praluent (alirocumab) significantly reduced LDL cholesterol. This analysis included 1,257 HeFH patients, the largest group of HeFH patients ever studied in a Phase III program. Results of this analysis were presented at the ESC Congress in September, and the 78 week results from two of the four trials included in the analysis, ODYSSEY FH I and II, were concurrently published online in the European Heart Journal.

The Phase III trial evaluating Synvisc-One in hip osteoarthritis did not reach its primary endpoint.

The FOCUS FH phase III study of Kynamro (mipomersen sodium) in patients with severe heterozygous familial hypercholesterolemia (severe HeFH) met its primary efficacy endpoint, a statistically significant reduction in LDL-cholesterol after 60 weeks of treatment of once weekly injections of 200 mg of Kynamro compared to placebo. However, the decision has been made not to move forward with the regulatory submission for severe HeFH in the U.S. Our efforts are focused on continuing to support patients with HoFH in the U.S.

Recruitment of the two Phase III studies evaluating the biosimilar insulin lispro has been completed.

Phase II:

Fluzone QIV HD (Quadrivalent high dose influenza vaccine) entered Phase II.
Sanofi has decided not to pursue development of vatelizumab, following the results of a Phase II pre-planned interim analysis in Multiple Sclerosis that revealed the primary efficacy endpoint was not met.
Sanofi has decided to out license the C-MET kinase inhibitor (SAR125844).

Phase I:

In October, Genzyme elected to opt into Alnylam’s investigational ALN-AT3 (SAR439774) hemophilia program for development and potential future commercialization in territories outside of North America and Western Europe. Genzyme retains its future opt-in right to co-develop and co-promote ALN-AT3 with Alnylam in North America and Western Europe. Specifically, Genzyme has the right to either co-develop and co-promote ALN-AT3 in Alnylam’s territory – with Alnylam maintaining development and commercialization control – or to maintain its RoW rights for ALN-AT3 and, if exercised by Genzyme, obtain a global license to ALN-AS1, Alnylam’s investigational RNAi therapeutic for the treatment of acute hepatic porphyrias. Genzyme will exercise this selection right upon completion of human proof-of-concept for the ALN-AS1 program, which is expected to occur in 2016.
An anti-miR21 RNA, SAR339375, entered Phase I in Alport syndrome.
An EP2 receptor agonist, SAR366234, entered Phase I in elevated intraocular pressure.
An anti-LAMP-1, SAR428926, entered Phase I in oncology.

A GLP-1R/GIPR dual agonist, SAR438335, entered Phase I in diabetes. Sanofi now has two dual agonists in Phase I in diabetes, a GLP1/GIPR and a GLP1-GCGR agonists.
2015 third-quarter and first 9-months 2015 financial results

Business Net Income(6)

In the third quarter of 2015, Sanofi generated net sales of €9,591 million, an increase of 9.2% on a reported basis (up 3.4% at constant exchange rates). Year-to-date sales were €27,779 million, an increase of 12.5% on a reported basis (up 3.6% at constant exchange rates).

Other revenues were €89 million, up 2.3% and €252 million, up 4.6% in the third quarter and the first nine months, respectively. At constant exchange rates, other revenues were down 8.0% in the third quarter and down 7.9% in the first nine months, reflecting lower royalties received on Enbrel sales in Europe.

In the third quarter, gross profit grew 11.3% (up 4.0% at constant exchange rates) to €6,682 million. The gross margin ratio improved by 1.3 percentage points to 69.7% versus the third quarter of 2014 under a favorable currency effect. Furthermore, positive impact from Genzyme and vaccine mix more than offset the negative impact of Lantus U.S. and Plavix generic competition in Japan. In the first nine months of 2015, the gross margin ratio was up 0.9 percentage points to 69.5% versus the first nine months of 2014. Sanofi continues to expect that the gross margin for 2015 will be around 69%.

Research and development expenses increased 18.2% (up 9.9% at constant exchange rates) to €1,355 million in the third quarter reflecting higher spend on dupilumab, the ODYSSEY cardiovascular outcome study with Praluent and the initiation of the new immuno-oncology alliance with Regeneron. Year-to-date R&D expenses increased 10.7% (up 2.6% at constant exchange rates) to €3,844 million. In the first nine months of 2015, the ratio of R&D to net sales was 0.3 percentage points lower at 13.8%.

Third-quarter selling and general expenses (SG&A) were up 12.2% to €2,461 million. At constant exchange rates, SG&A was up 6.2% mainly reflecting the launch costs in North-America of Praluent, the Toujeo Direct-to-Consumer advertising in the U.S. and commercial expenses supporting the Multiple Sclerosis franchise and Animal Health. The ratio of SG&A to net sales increased 0.7 percentage points to 25.7% compared with the third quarter of 2014. Year-to-date SG&A expenses increased 15.6% to €7,547 million, (up 6.2% at constant exchange rates). In the first nine months of 2015, the ratio of selling and general expenses to net sales was 0.8 percentage points higher to 27.2% compared with the first nine months of 2014.

Other current operating income net of expenses was -€136 million in the third quarter versus €39 million in the third quarter of 2014 which included a €40 million capital gain associated with the termination of a license in the U.S. In the third quarter, Sanofi recorded €137 million as a foreign exchange loss with respect to its subsidiaries based in Venezuela, mainly resulting from the re-measurement of intra-Group USD denominated payables, using the expected foreign exchange rate applicable for the future settlement of those payables. As of 30 September 2015, the total foreign exchange loss on Venezuela was €237 million. Other current operating income net of expenses was -€223 million in the first nine months of 2015 versus €68 million in the same period of 2014.

The share of profits from associates was €78 million in the third quarter versus €43 million in the third quarter of 2014. This included Sanofi’s share in Regeneron profit recorded under the equity method since the beginning of April 2014 as well as Sanofi’s share of profit in Sanofi Pasteur MSD (the Vaccines joint venture with Merck & Co. in Europe). In the first nine months, the share of profits from associates was €139 million versus €82 million for the same period of 2014.

Non-controlling interests were -€25 million in the third quarter versus -€31 million in the third quarter of 2014. Year-to-date non-controlling interests were -€87 million versus -€96 million for the same period of 2014.

Third-quarter business operating income(7) was €2,783 million, up 2.5%. At constant exchange rates, business operating income was down 0.4%. The ratio of business operating income to net sales was 1.9 percentage points lower to 29.0% versus the same period of last year. Year-to-date business operating income increased 10.6% to €7,747 million (up 1.9% at constant exchange rates).

In the first nine months of 2015, the ratio of business operating income to net sales decreased by 0.5 percentage points to 27.9%.

Net financial expenses were €105 million in the third quarter compared to €139 million in the third quarter of 2014. Year-to-date net financial expenses were €314 million versus €309 million in the first nine months of 2014.

The full-year effective tax rate forecast has been reviewed at 24% (previously 25%), consequently the third quarter effective tax rate was 22.2%.

Third-quarter business net income(6) increased 8.3% to €2,096 million (up 5.0% at constant exchange rates). The ratio of business net income to net sales was down slightly (0.1 percentage point) to 21.9% compared with third quarter of 2014. Year-to-date business net income was up 12.8% to €5,662 million, (up 3.7% at constant exchange rates). The ratio of business net income to net sales improved by 0.1 percentage points to 20.4% compared to the first nine months of 2014.

In the third quarter of 2015, business earnings per share(6) (EPS) was €1.61, an increase of 9.5% on a reported basis and 6.1% at constant exchange rates. The average number of shares outstanding was 1,305.5 million in the third quarter versus 1,313.0 million in the same period in 2014. In the first nine months of 2015, business earnings per share(6) was €4.33, up 13.6% on a reported basis and up 4.5% at constant exchange rates. The average number of shares outstanding was 1,306.6 million in the first nine months versus 1,315.8 million in the first nine months of 2014.
(6) See Appendix 8 for definitions of financial indicators, and Appendix 3 for reconciliation of business net income to IFRS net income reported
(7) Business operating income is the segment result used by the Group. The consolidated income statement for Q3 2015 is provided in Appendix 4

From business net income to IFRS net income reported (see Appendix 3)

In the first nine months of 2015, the main reconciling items between business net income and IFRS net income reported were:

A €1,827 million amortization charge related to fair value remeasurement on intangible assets of acquired companies (primarily Aventis: €493 million, Genzyme: €666 million and Merial: €385 million) and to acquired intangible assets (licenses/products: €95 million). A €598 million amortization charge on intangible assets related to fair value remeasurement of acquired companies (primarily Aventis: €139 million, Genzyme: €217 million and Merial: €144 million), and to acquired intangible assets (licenses/products: €38 million) was recorded in the third quarter. These items have no cash impact on the Group.

An impairment of intangible assets of €237 million (of which €209 million in the third quarter of 2015 mainly linked to Synvisc and vatelizumab). This item has no cash impact on the Group.

An income of €161 million mainly reflecting a decrease in the fair value of contingent considerations related to the CVRs (€127 million, of which an income of €109 million in the third quarter of 2015) and a decrease of Bayer contingent considerations (€20 million, of which a charge of €19 million in the third quarter of 2015) linked to Lemtrada.

Restructuring costs of €439 million (including €58 million in the third quarter mainly related to transformation in Europe and Venezuela).

A €871 million tax effect arising from the items listed above, comprising €641 million of deferred taxes generated by amortization charged against intangible assets, €150 million associated with restructuring costs, €87 million associated with impairment of intangible assets and a charge of €7 million associated with fair value remeasurement of contingent consideration liabilities The third quarter tax effect was €310 million, including €210 million of deferred taxes generated by amortization charged against intangible assets and a charge of €77 million associated with fair value remeasurement of contingent consideration liabilities (see Appendix 3).
A tax of €111 million on dividends paid to shareholders of Sanofi.

In "Share of profits/losses from associates", a charge of €132 million, net of tax, (of which €5 million in the third quarter of 2015) mainly relating to the share of the fair-value re-measurements on assets and liabilities as part of the acquisition of associates and to the share of amortization of intangible assets of joint-ventures. This item has no cash impact on the Group.

TESARO Announces Third-Quarter 2015 Operating Results

On October 29, 2015 TESARO, Inc. (NASDAQ:TSRO), an oncology-focused biopharmaceutical company, reported operating results for third-quarter 2015 and provided an update on the Company’s development programs (Press release, TESARO, OCT 29, 2015, View Source [SID:1234507845]).

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"The FDA approval of TESARO’s first product, VARUBI, offers a new treatment option for patients with cancer who are affected by nausea and vomiting caused by chemotherapy and represents a significant milestone for TESARO," said Lonnie Moulder, CEO of TESARO. "Our field organization is fully in place, and we look forward to providing VARUBI to patients in mid-November. In addition to VARUBI, we are building a franchise around niraparib in ovarian cancer, and we are enthusiastic about the potential to expand our development program for this molecule to include several new tumor types. The Phase 3 NOVA trial of niraparib was initiated more than two years ago, and patient enrollment completed seven months ago. Based upon a recently completed HRD assessment of tumor samples and a greater than anticipated duration of treatment, we now look forward to top-line data from NOVA in the second quarter of 2016. We are very optimistic about the potential of niraparib for patients with ovarian, breast and other cancers."

Recent Business Highlights

On September 1, 2015, the U.S. Food and Drug Administration (FDA) approved VARUBI (oral rolapitant), in combination with other antiemetic agents in adults, for the prevention of delayed nausea and vomiting associated with initial and repeat courses of emetogenic cancer chemotherapy, including, but not limited to, highly emetogenic chemotherapy.

The National Comprehensive Cancer Network (NCCN) added VARUBI to the NCCN Clinical Practice Guidelines in Oncology (NCCN Guidelines) Antiemesis Version 2.2015 as a recommended option, in combination with other antiemetic agents, for patients receiving both high emetic risk intravenous chemotherapy (HEC) and moderate emetic risk intravenous chemotherapy (MEC). Category 1, the highest level category of evidence and consensus, was granted to rolapitant for both HEC and MEC chemotherapy.

The TESARO field organization is now over 120 associates strong and includes sales management, area managers, corporate account directors, medical science liaisons, and clinical nurse educators. Preparation is ongoing to support the successful U.S. commercial launch of VARUBI in mid-November.

The planned intravenous (IV) rolapitant clinical program is now complete, and following a pre-NDA meeting with the U.S. FDA, a New Drug Application (NDA) will be submitted.

An assessment of the patient tumor samples collected from patients enrolled in the Phase 3 NOVA trial of niraparib was recently completed using the myChoice HRD test in preparation for progression-free survival (PFS) endpoint analysis. As anticipated, results from this testing determined that approximately 50% of patients enrolled in the non-gBRCA cohort have HRD-positive tumors.

Based on the observed event rate, new estimates for the NOVA timing of PFS events indicate that top-line PFS results for NOVA are now expected to be available in Q2 2016.

Enrollment of the QUADRA trial of niraparib for the treatment of patients with ovarian cancer who have received three or more prior lines of chemotherapy is now more than 50 percent complete.

Antibody drug candidates targeting PD-1, TIM-3, and LAG-3 continue to advance, and Investigational New Drug (IND) application preparations are underway for TSR-042 and TSR-022, our anti-PD-1 and anti-TIM-3 antibody candidates.
The Phase 1/2 clinical trial of TSR-011 has been discontinued, and resources are being reprioritized to support development programs for niraparib and our immuno-oncology candidates.

Third Quarter 2015 Financial Results

TESARO reported a net loss of $66.6 million, or ($1.66) per share, for the third quarter of 2015, compared to a net loss of $36.2 million, or ($1.01) per share, for the third quarter of 2014.

Research and development expenses increased to $40.1 million for the third quarter of 2015, compared to $29.9 million for the third quarter of 2014, driven primarily by higher costs related to expanded development activities and increased headcount.
Selling, general, and administrative expenses increased to $22.8 million for the third quarter of 2015, compared to $6.3 million for the third quarter of 2014, primarily due to pre-launch commercial activities in support of VARUBI, increased commercial headcount, and higher professional service fees.

Operating expenses, as described above, include total non-cash, stock-based compensation expense of $8.1 million for the third quarter of 2015, compared to $2.9 million for the third quarter of 2014.

As of September 30, 2015, TESARO had approximately $302.5 million in cash and cash equivalents and approximately 40.0 million outstanding shares of common stock. TESARO expects cash utilization to be in the mid- to high-$50 million range for the fourth quarter of 2015, excluding a $15 million milestone payment that will be due upon the first commercial sale of VARUBI, which is expected to occur in November.

Corporate Objectives

TESARO anticipates achieving the following key objectives:

Launch VARUBI into the U.S. market in mid-November 2015;
Submit the NDA for IV rolapitant in Q1 2016;
Submit the oral rolapitant Marketing Authorization Application (MAA) to the European Medicines Agency (EMA) in Q2 2016;
Report top-line data from the Phase 3 NOVA trial of niraparib in Q2 2016;
Report top-line data from the QUADRA trial of niraparib in Q2 2016;
Submit the niraparib NDA in 2H 2016;
Continue to enroll the Phase 3 BRAVO trial of niraparib in breast cancer patients with germline BRCA mutations through 2016;
Initiate enrollment in the niraparib/KEYTRUDA (pembrolizumab) combination trial in Q1 2016;
Initiate enrollment in the Phase 3 clinical trial of niraparib in first line ovarian cancer (PRIMA) in Q1 2016;
Advance the development of TSR-042 (anti-PD-1 antibody) to support submission of an IND application to the U.S. FDA at year-end 2015; and
Advance the IND-enabling studies for TSR-022 (anti-TIM-3 clinical candidate) to support submission of an IND application in Q2 2016.

Varian Medical Systems Reports Results for Fourth Quarter of Fiscal Year 2015

On October 28, 2015 Varian Medical Systems (NYSE:VAR) reported non-GAAP net earnings of $1.04 per diluted share and GAAP earnings of $0.99 per diluted share for the fourth quarter of fiscal year 2015 (Press release, Varian Medical Systems, OCT 28, 2015, View Source [SID:1234507824]). For the full fiscal year 2015, non-GAAP earnings were $4.29 per diluted share, and GAAP earnings were $4.09 per diluted share. Varian’s revenues totaled $818 million for the fourth quarter of fiscal year 2015, up 1 percent from the year-ago quarter and up 6 percent in constant currency. Varian’s revenues for the full fiscal year were $3.1 billion, up 2 percent versus fiscal year 2014 and up 6 percent in constant currency. The company ended the fourth quarter with a $3.5 billion backlog, up 10 percent from the end of fiscal year 2014.

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"During the quarter, our Oncology Systems business generated healthy constant currency order growth, the Particle Therapy business gathered momentum, and the Imaging Components business continued to experience declines in orders, revenues and margins," said Dow R. Wilson, CEO of Varian Medical Systems. "As we previously reported, we experienced a shortfall of high-margin revenues in our Oncology business when several TrueBeam systems and related software slipped out of the quarter."

The company finished the fiscal year with $845 million in cash and cash equivalents and $496 million of debt. Cash flow from operations was $153 million for the fourth quarter and $470 million for the fiscal year. During the quarter, the company spent $128 million to repurchase about 1.5 million shares of common stock.

Oncology Systems

Oncology Systems’ fourth quarter revenues totaled $633 million, up 2 percent from the same quarter of fiscal year 2014 and up 9 percent in constant currency. Annual revenues were $2.3 billion, even with the prior fiscal year, and up 6 percent in constant currency.

Fourth-quarter gross orders were $919 million, equal to the year-ago quarter and up 5 percent in constant currency. In the Americas, fourth quarter Oncology gross orders declined by 5 percent in dollars and constant currency. In EMEA, gross orders were up 13 percent in dollars and up 25 percent in constant currency. In APAC, gross orders declined by 3 percent in dollars but rose 6 percent in constant currency. Annual Oncology gross orders were $2.7 billion, even with fiscal year 2014 and up 6 percent in constant currency. In the Americas, annual gross orders were up 1 percent in dollars and constant currency. In EMEA gross orders were flat in dollars but up 12 percent in constant currency. In APAC, order growth was also flat in dollars but up 9 percent in constant currency.

"Oncology gross orders were strong in EMEA during the quarter when we booked orders for over 100 systems," said Wilson. "North American orders grew by 4 percent in the quarter driven by customers continuing to upgrade to newer technologies, replacements of competitors’ products, and increased software sales. We believe we gained share in constant currency in all regions."

Imaging Components

Imaging Components revenues were $155 million for the fourth quarter, down 8 percent from the year-ago period, and $611 million for the fiscal year, down 7 percent from fiscal year 2014. Gross orders were $165 million for the fourth quarter, down 30 percent from the year-ago period, and totaled $605 million for the fiscal year, down 16 percent from fiscal year 2014.

"Price erosion in response to aggressive euro- and yen-based competitors was the principal cause of the decline in orders and revenues for panels and tubes in our Imaging Components business," said Wilson. "Gross orders for security products were down $63 million or 57 percent for the fiscal year, and annual revenues fell by $34 million or 37 percent, due largely to instability in key international markets. The company has initiated a restructuring program to right-size the Imaging Components business and to get it back on a growth track."

During the fourth quarter of fiscal year 2015, the company paid approximately €52 million in cash to acquire Claymount Investments B.V., a privately-held, Netherlands-based supplier of components and subsystems for X-ray imaging equipment manufacturers.

Other

The company’s Other category, including the Varian Particle Therapy business and the Ginzton Technology Center, recorded revenues of $30 million for the fourth quarter and $144 million for fiscal year 2015. It generated gross orders of $141 million in the quarter and $317 million for the fiscal year. During the quarter, the Particle Therapy business booked orders for three proton therapy centers, comprising two in the UK and one in New York. "It is gratifying to see growing global market demand for Varian’s proton therapy systems," said Wilson. "We are gaining momentum in this important clinical space."

Outlook

"We believe that for fiscal year 2016 total company non-GAAP earnings will be in the range of $4.45 to $4.55 per diluted share and revenues will increase by about 4 to 5 percent on a reported basis," said Wilson. "For the first quarter of fiscal year 2016, we expect revenues to be roughly even with the year-ago quarter in dollars. With ongoing challenges experienced by Imaging Components in the second half of fiscal year 2015 as well as the effect of year-over-year changes in currency exchange rates, we expect non-GAAP earnings for the first quarter of fiscal year 2016 to be in the range of $0.88 to $0.92 per diluted share."

Non-GAAP Items

Beginning this quarter, the company is reporting non-GAAP operating earnings, non-GAAP net earnings and non-GAAP diluted earnings per share to provide comparisons against prior periods excluding certain items that may not be indicative of its core operating results and business outlook, allow better comparability among company peers, and provide additional transparency. Non-GAAP operating earnings and non-GAAP net earnings exclude the following items that are included under GAAP: amortization of intangible assets, acquisition-related expenses and or benefits, restructuring charges, impairment charges, significant litigation charges or benefits and associated legal costs. From time to time, the company may exclude other items if it is consistent with the goal of providing useful information to investors. Tax effects on non-GAAP items are calculated based on the company’s effective tax rate other than when the underlying item has a materially different tax treatment. Additional details and a table reconciling the GAAP to non-GAAP financial measures are included in this release.