Innovent Announces Oral Presentations at ESMO Plenary and ESMO GI Congress on Clinical Data of IBI363 (PD-1/IL-2) and IBI343 (CLDN18.2 ADC)

On May 19, 2024 Innovent Biologics, Inc. ("Innovent") (HKEX: 01801), a world-class biopharmaceutical company that develops, manufactures and commercializes high quality medicines for the treatment of oncology, cardiovascular and metabolic, autoimmune, ophthalmology and other major diseases, reported that the company will deliver oral presentations on clinical data of its first-in-class PD-1/IL-2 bispecific antibody fusion protein (R&D code: IBI363) and novel Topoi anti-Claudin18.2 ADC (R&D code: IBI343) at the upcoming medical conferences in June, including ESMO (Free ESMO Whitepaper) Virtual Plenary and ESMO (Free ESMO Whitepaper) Gastrointestinal Cancers Congress (ESMO GI) 2024. Details are as follows (Press release, Innovent Biologics, MAY 19, 2024, View Source [SID1234643430]):

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ESMO Virtual Plenary, June 13-June 14, 2024

Title: First-in-class PD-1/IL-2 bispecific antibody fusion protein IBI363 in patients (pts) with advanced solid tumors: First-in-human phase I study
Presentation Form: Oral
Presentation Time: 13 Jun 2024 18:30-19:30 CEST & 14 June 2024 13:00-14:10 CEST
Presenting Author: Prof. Xueli Bai, The first affiliated hospital, Zhejiang University School of Medicine

ESMO Gastrointestinal Cancers Congress, June 26-June 29, 2024, Munich, Germany

Title: Anti-claudin 18.2 (CLDN18.2) antibody-drug conjugate (ADC) IBI343 in patients (pts) with solid tumors and gastric/gastro-esophageal junction adenocarcinoma (G/GEJ AC): A phase 1 study
Publication Number: 396MO
Presentation Form: Oral
Presentation Time: 29 June 2024 08:45-10:00 CEST
Presenting Author: Jia (Jenny) Liu, St Vincent’s Hospital Sydney

Dr. Hui Zhou, Senior Vice President of Innovent, stated: "We will present a robust set of clinical data for our next-generation innovative bispecific antibodies and ADC molecules at multiple conferences in the near term. We observed the preliminary efficacy and safety signals for those innovative candidates, underscoring their potential for further development and clinical value. Innovent leverages our world-class antibody-based platform, differentiated ADC technology and deep scientific understanding to build the new generation innovative pipeline of "IO+ADC". We strive to solve the unmet needs of existing therapies and fill the treatment gap for cancer patients worldwide."

CiMaas and CYTEA BIO are pleased to announce their collaboration on Natural Killer cells

On May 19, 2024 CiMaas reported that it will provide CYTEA BIO with the GMP-grade K562-F012 feeder cells for the expansion of its umbilical cord blood-derived NK cells (Press release, CiMaas, MAY 19, 2024, View Source [SID1234643429]). Conversely, CYTEA BIO will supply CiMaas with Pin antibodies for the pre-arming of CiMaas NK cells to assess the benefit it brings and the opportunity to pursue a longer-term partnership.

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CYTEA BIO is a Swiss/French biotech company dedicated to developing cell therapeutics using its patented Pin platform. This unique approach allows pre-arming Fc-engineered targeting ligands onto genetically unmodified effector cells to orientate and harness a naturally occurring cytotoxicity process. With this platform, an infinite number of products can be envisaged, with ligands and/or effector cells being interchanged. Pre-arming human allogeneic NK cells with Fc-Engineered antibodies (PinTM antibodies) highlighted the power of this strategy, improving the functional and targeted cytotoxicity of the NK cells against various cancer models. CYTEA BIO has initiated a lead development program using pre-armed human allogeneic NK cells with Pin anti-EGFR antibody for the treatment of glioblastoma multiforme.

Ono Receives Approvals of BRAFTOVI® and MEKTOVI® for Expanded Use for Two New Indications in Japan

On May 17, 2024 Ono Pharmaceutical Co., Ltd. reported that it has received supplemental approvals for BRAFTOVI (generic name: encorafenib) Capsule ("BRAFTOVI"), a BRAF inhibitor, and MEKTOVI (generic name: binimetinib) Tablet ("MEKTOVI"), a MEK inhibitor, when used in combination, in Japan for the two new indications of "unresectable thyroid cancer with a BRAF mutation that has progressed following chemotherapy", and "unresectable anaplastic thyroid cancer with a BRAF mutation" (Press release, Ono, MAY 17, 2024, View Source [SID1234646254]).

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 These approvals are based on the results of a Phase 2 study (ONO-7702/7703-03), conducted in Japan in 22 patients with unresectable BRAFV600-mutant thyroid cancer, including 5 patients with anaplastic thyroid cancer. The study met its primary endpoint of objective response rate (ORR) as assessed by the Independent Central Review in the overall patient population, which was 54.5% (12/22 cases, 95% confidence interval: 32.2 – 75.6%) in the combination therapy of BRAFTOVI and MEKTOVI. The safety profile of the combination therapy of BRAFTOVI and MEKTOVI in the study was consistent with those previously reported in the clinical trials of BRAFTOVI and MEKTOVI.

About Phase 2 study (ONO-7702/7703-03)
 The study is a multi-centre, open-label, uncontrolled Phase 2 study (ONO-7702/7703-03), conducted in Japan, evaluating the efficacy and safety of the combination therapy of BRAFTOVI and MEKTOVI in patients with unresectable BRAFV600-mutant thyroid cancer. Patients received the combination therapy with BRAFTOVI 450 mg once daily, and MEKTOVI 45 mg twice daily, until it was determined that treatment could not be given due to disease progression or safety reasons. The primary endpoint of the study was objective response rate (ORR) as assessed by the Independent Central Review. Secondary endpoints include ORR as assessed by physician of each medical institutes, disease control rate (DCR), overall survival (OS) and progression-free survival (PFS).

About Thyroid Cancer
 Thyroid cancer (TC) is a malignant tumor that develops in the thyroid tissue located around the trachea or in front of the neck. Histologically, it is roughly divided into differentiated carcinoma (approximately 97% of TC), undifferentiated carcinoma (1 – 2%), and medullary carcinoma (1 – 2%). In Japan, it is estimated that approximately 18,700 new cases are diagnosed with TC per year with approximately 1,900 deaths per year resulting from the disease in 2023*. BRAF mutation is reported in 37 – 68% of TC patients.

Cancer Statics in Japan, 2024, The Editorial Board of Cancer Statistics, Foundation for Promotion of Cancer Research (FPCR), March 2024

Overview of BRAFTOVI Capsule 50 mg and 75 mg
Product Name BRAFTOVI Capsule 50 mg and 75 mg
Generic name (JAN) Encorafenib
Indication
Unresectable melanoma with a BRAF mutation
Unresectable advanced or recurrent colorectal cancer with a BRAF mutation that has progressed following chemotherapy
Unresectable thyroid cancer with a BRAF mutation that has progressed following chemotherapy
Unresectable anaplastic thyroid cancer with a BRAF mutation
Dosage and administration

In combination with binimetinib, usually, for adults, administer 450 mg of encorafenib orally once a day. According to patients’ condition, the dose should be reduced.

In combination with cetuximab (genetical recombination) or with binimetinib and cetuximab (genetical recombination), usually, for adults, administer 300 mg of encorafenib orally once a day. According to patients’ condition, the dose should be reduced.

Manufacturer/distributor Ono Pharmaceutical Co., Ltd.
Note: Underlined parts show the revised ones due to this approval.

Overview of MEKTOVI Tablet 15 mg
Product Name MEKTOVI Tablet 15 mg
Generic name (JAN) Binimetinib
Indication
Unresectable melanoma with a BRAF mutation
Unresectable advanced or recurrent colorectal cancer with a BRAF mutation that has progressed following chemotherapy
Unresectable thyroid cancer with a BRAF mutation that has progressed following chemotherapy
Unresectable anaplastic thyroid cancer with a BRAF mutation
Dosage and administration

In combination with encorafenib, usually, for adults, administer 45 mg of encorafenib orally twice a day. According to patients’ condition, the dose should be reduced.

In combination with encorafenib and cetuximab (genetical recombination), usually, for adults, administer 45 mg of binimetinib orally twice a day. According to patients’ condition, the dose should be reduced.

Manufacturer/distributor Ono Pharmaceutical Co., Ltd.
Note: Underlined parts show the revised ones due to this approval.

About BRAFTOVI and MEKTOVI
 BRAFTOVI is a small molecule BRAF kinase inhibitor and MEKTOVI is a small molecule MEK inhibitor. BRAF and MEK are important protein kinases in the MAPK signalling pathway (RAS-RAF-MEK-ERK), which regulates several key cellular activities including proliferation, differentiation, survival and angiogenesis. Inappropriate activation of proteins in this pathway has been shown to occur in many types of cancers including melanoma, colorectal cancer and thyroid cancer. Both BRAFTOVI and MEKTOVI target key enzymes in this pathway.
 In Japan, Ono received a manufacturing and marketing approval of BRAFTOVI and MEKTOVI for the treatment of unresectable melanoma with a BRAF mutation in combination therapy of the products in January 2019 and launched them in February 2019. Thereafter, Ono received additional approval in November 2020 for the treatment of unresectable advanced or recurrent colorectal cancer with a BRAF mutation that has progressed following chemotherapy, in triplet combination treatment of BRAFTOVI, MEKTOVI and cetuximab, an anti-human EGFR monoclonal antibody, as well as in doublet combination treatment of BRAFTOVI and cetuximab.
 Abroad, Array BioPharma Inc. (a wholly owned subsidiary of Pfizer Inc.) and its collaboration partner, Pierre Fabre, received an approval of BRAFTOVI and MEKTOVI for the treatment of unresectable or metastatic melanoma with BRAFV600E or V600K mutation and launched them in 2018 in the US and EU, respectively. Thereafter, the companies received supplemental approval for the treatment of metastatic colorectal cancer with a BRAFV600E mutation following prior therapy in the US and EU in 2020. Additionally, Pfizer received supplemental approval in the US for the treatment of metastatic non-small cell lung cancer with a BRAFV600E mutation in 2023.

About the Ono Pharmaceutical Co., Ltd. and Pfizer Inc. Collaboration
 In May 2017, Ono entered into the license agreement with Array BioPharma Inc. (became a subsidiary of Pfizer Inc. as of July 30, 2019) regarding BRAFTOVI (encorafenib), a BRAF inhibitor and MEKTOVI (binimetinib), a MEK inhibitor and received rights to develop and commercialize both products in Japan and South Korea.

Autolus Therapeutics Reports First Quarter 2024 Financial Results and Business Updates

On May 17, 2024 Autolus Therapeutics plc (Nasdaq: AUTL), a clinical-stage biopharmaceutical company developing next-generation programmed T cell therapies, reported its operational and financial results for the first quarter ended March 31, 2024 (Press release, Autolus, MAY 17, 2024, View Source [SID1234643422]).

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"We continue to engage with the FDA in the regulatory review process for obecabtagene autoleucel (obe-cel) in adult ALL as we head towards the PDUFA target action date of November 16, 2024, and are driving commercial readiness activities across the Company," said Dr. Christian Itin, Chief Executive Officer of Autolus. "We’re also delighted that our abstracts from the pivotal FELIX Phase 2 trial have been accepted for oral presentations at ASCO (Free ASCO Whitepaper) and EHA (Free EHA Whitepaper) this year and we look forward to sharing further long-term data and additional subset analyses."

"In addition, the first two patients have been enrolled into our dose confirmation trial (CARLYSLE) of obe-cel in Systemic Lupus Erythematosus (SLE) and the study is on track for initial data by end of 2024."

Key obe-cel updates and anticipated milestones:

Obe-cel in relapsed / refractory (r/r) adult B-cell Acute Lymphoblastic Leukemia (ALL) – The FELIX Study
Obe-cel Biologics License Application (BLA) for r/r B-ALL submitted to the FDA in November 2023; PDUFA target action date of November 16, 2024. A marketing authorization application (MAA) to the European Medicines Agency (EMA) was accepted in April 2024. For the UK we are evaluating a filing based on an international recognition procedure.
Pooled analysis of the FELIX Phase 1b/2 study presented at ASH (Free ASH Whitepaper) in December 2023 demonstrated prolonged event free survival and low overall immunotoxicity across all cohorts in r/r B-ALL, and particularly in patients with low leukemic burden at lymphodepletion.
Further long-term data from the FELIX study including additional subset analysis will be presented in oral and poster presentations at the American Society of Clinical Oncology (ASCO) (Free ASCO Whitepaper) annual meeting (ASCO – May 31 – June 4, 2024), and European Hematology Association (EHA) (Free EHA Whitepaper) congress (EHA – June 13 – 16, 2024) respectively.
Obe-cel in B-cell mediated autoimmune diseases
The Phase 1 dose confirmation study (CARLYSLE) in refractory systemic lupus erythematosus (SLE) patients is ongoing. Two patients have been enrolled and Autolus continues to expect initial clinical data in late 2024.
Pipeline clinical trials, in collaboration with University College London (UCL), updates and anticipated milestones:

AUTO8 in Multiple Myeloma – Phase 1 MCARTY Study
AUTO8 is a next-generation product candidate for multiple myeloma, which includes two CARs for the multiple myeloma targets, BCMA and CD19. Initial data from the MCARTY Phase 1 study in multiple myeloma presented at ASH (Free ASH Whitepaper) in December 2023 showed AUTO8 was well tolerated, with responses observed in all patients. Enrollment of the initial cohorts are complete and further updates from the MCARTY study are anticipated in H2 2024.
AUTO6NG in Neuroblastoma – Phase 1 MAGNETO Study
AUTO6NG contains a CAR that targets GD2 alongside additional programming modules to enhance the activity and persistence. A Phase 1 clinical study in children with r/r neuroblastoma was opened for enrollment in the fourth quarter of 2023.
Strategic developments:

In February 2024, BioNTech and Autolus announced a strategic CAR T cell therapy collaboration to advance their pipelines and expand late-stage programs, for $50 million cash upfront and up to $582 million in potential option exercise and milestone payments. Additionally, Autolus sold $200 million of ADSs to BioNTech in a concurrent private placement financing transaction.
In February 2024, Autolus completed an underwritten offering in the United States at a price of $6.00 per ADS, for total gross proceeds of $350 million before underwriting fees and offering expenses.
Operational Updates:

In March 2024, The Nucleus manufacturing facility in Stevenage obtained a Manufacturer’s Importation Authorization (MIA), together with the accompanying GMP certificate. This authorization enables Autolus to manufacture products for global commercial and clinical supply at The Nucleus, effective as of March 18, 2024.
In April 2024, Autolus announced that the European Medicines Agency (EMA) had accepted its Marketing Authorization Application (MAA) for obe-cel for patients with relapsed/refractory (r/r) adult B-cell Acute Lymphoblastic Leukemia (ALL). The MAA submission was based on data from the pivotal Phase 2 FELIX study of obe-cel in adult r/r B-ALL.
In April 2024, Autolus entered into a distribution services agreement with a subsidiary of Cardinal Health to support the ordering and distribution of obe-cel in the United States, following the receipt of regulatory approval.
In April 2024, Autolus announced the appointment of Mike Bonney as Chairman of the Board, and Ravi Rao M.D., as Non-Executive Director. John H. Johnson advised the Board of his decision to step down from his role as Chairman of the Board and Non-Executive Director, effective April 1, 2024.
Scientific Publications:

In January 2024, Autolus announced the publication of a paper in ACS Chemical Biology entitled: ‘Designer small molecule control system based on Minocycline induced disruption of protein-protein interaction’ – Jha et al., ACS Chemical Biology (2024) doi:10.1021/acschembio.3c00521; [Link]
In February 2024, Autolus announced the publication of a paper in Nature Communications entitled: ‘Structure-Guided Engineering of Immunotherapies Targeting TRBC1 and TRBC2 in T Cell Malignancies’ – Ferrari et al., Nat Commun 15, 1583 (2024) doi:10.1038/s41467-024-45854-3; [Link]
In March 2024, Autolus announced the publication of a paper in Blood Cancer Journal entitled: ‘Dual T-cell constant β chain (TRBC)1 and TRBC2 staining for the identification of T-cell neoplasms by flow cytometry – Horna et al., Blood Cancer J. 14, 34 (2024) doi: 10.1038/s41408-024-01002-0; [Link]
2024 Expected News Flow:

Obe-cel FELIX data update at ASCO (Free ASCO Whitepaper), EHA (Free EHA Whitepaper) & ASH (Free ASH Whitepaper) May, June & Dec 2024
Obe-cel Marketing Authorization Application to MHRA Second half 2024
Obe-cel U.S. FDA PDUFA target action date November 16, 2024
Obe-cel in autoimmune disease – initial data from SLE Phase 1 study Late 2024

Financial Results (Unaudited) for the Quarter Ended March 31, 2024

Cash and cash equivalents at March 31, 2024, totaled $758.5 million, as compared to $239.6 million at December 31, 2023.

Total operating expenses, net for the three months ended March 31, 2024, were $38.8 million, as compared to $39.1 million, for the same period in 2023.

Research and development expenses increased from $27.4 million to $30.7 million for the three months ended March 31, 2024, compared to the same period in 2023. This change was primarily due to increases in operating costs related to the Company’s new commercial manufacturing facility, employee salaries and related costs, clinical trial costs related to obe-cel, and a decrease in our U.K. reimbursable R&D tax credits claimable through the U.K. small and medium-sized entity (SME) scheme. These were partially offset by decreases in professional consulting fees, legal fees, manufacturing costs related to obe-cel clinical supply, information technology infrastructure fees and general office expenses.

General and administrative expenses increased from $9.3 million to $18.2 million for the three months ended March 31, 2024, compared to the same period in 2023. This increase was primarily due to salaries and other employment-related costs driven by an increase in general and administrative headcount supporting the overall growth of the business, primarily relating to pre-commercialization activities.

Net loss was $52.7 million for the three months ended March 31, 2024, compared to $39.8 million for the same period in 2023. The basic and diluted net loss per ordinary share for the three months ended March 31, 2024, totaled $(0.24), compared to a basic and diluted net loss per ordinary share of $(0.23) for 2023.

Autolus estimates that, with its current cash and cash equivalents and proceeds received from the strategic alliance with BioNTech and the private placement and underwritten equity financing, it is well capitalized to drive the full launch and commercialization of obe-cel in r/r adult ALL as well as to advance its pipeline development plans, which includes providing runway to data in the first pivotal study of obe-cel in autoimmune disease.

Financial Results for the Quarter Ended March 31, 2024
Selected Unaudited Condensed Consolidated Balance Sheet Data
(In thousands)

March 31 December 31
2024 2023
Assets
Cash and cash equivalents $ 758,529 $ 239,566
Total current assets $ 804,298 $ 275,302
Total assets $ 901,436 $ 375,381
Liabilities and shareholders’ equity
Total current liabilities $ 43,985 $ 44,737
Total liabilities $ 319,406 $ 263,907
Total shareholders’ equity $ 582,030 $ 111,474

Selected Unaudited Condensed Consolidated Statements of Operations and Comprehensive Loss Data
(In thousands, except share and per share amounts)

Three Months Ended March 31,
2024 2023
License revenues $ 10,091 $ 1,292
Operating expenses:
Research and development (30,671 ) (27,388 )
General and administrative (18,177 ) (9,284 )
Loss on disposal of property and equipment - (3,768 )
Total operating expenses, net (38,757 ) (39,148 )
Total other expenses, net (13,941 ) (677 )
Net loss before income tax (52,698 ) (39,825 )
Income tax benefit 8 14
Net loss (52,690 ) (39,811 )
Other comprehensive income (loss):
Foreign currency exchange translation adjustment 58 5,641
Total comprehensive loss $ (52,632 ) $ (34,170 )

Basic and diluted net loss per ordinary share $ (0.24 ) $ (0.23 )
Weighted-average basic and diluted ordinary shares 222,170,707 173,825,825

Conference Call
Management will host a conference call and webcast at 08:30 am EDT/13:30 pm BST to discuss the Company’s financial results and provide a general business update. Conference call participants should pre-register using this link to receive the dial-in numbers and a personal PIN, which are required to access the conference call.

A simultaneous audio webcast and replay will be accessible on the events section of Autolus’ website.

Ultragenyx Reports Inducement Grant Under Nasdaq Listing Rule 5635(c)(4)

On May 17, 2024 Ultragenyx Pharmaceutical Inc. (NASDAQ: RARE), a biopharmaceutical company focused on the development and commercialization of novel therapies for rare and ultrarare diseases, reported the grant of 17,180 restricted stock units of the company’s common stock to ten newly hired non-executive officers of the company (Press release, Ultragenyx Pharmaceutical, MAY 17, 2024, View Source [SID1234643427]). The awards were approved by the compensation committee of the company’s board of directors and granted under the Ultragenyx Employment Inducement Plan, with a grant date of May 16, 2024, as an inducement material to the new employees entering into employment with Ultragenyx in accordance with Nasdaq Listing Rule 5635(c)(4).

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The restricted stock units vest over four years, with 25% of the underlying shares vesting on each anniversary of the grant date, subject to the employee being continuously employed by the company as of such vesting dates.