Medigene to Present Expitope 3.0 at the 20th Annual Meeting of the Association for Cancer Immunotherapy (CIMT)

On April 27, 2023 Medigene AG (Medigene, FSE: MDG1, Prime Standard), an immuno-oncology platform company focusing on the discovery and development of T cell immunotherapies for solid tumors, reported that it will be presenting at the 20th Association for Cancer Immunotherapy (CIMT) (Free CIMT Whitepaper) annual meeting being held on May 3-5, 2023, in Mainz (Press release, MediGene, APR 27, 2023, View Source [SID1234630629]).

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The data to be presented will focus on Expitope 3.0, an in silico tool to identify immunogenic epitopes as suitable T cell receptor (TCR) target specificities. Moreover, Expitope 3.0, enables the comparison of expression of epitopes in various healthy tissues to predict potential cross-reactivity and off-target toxicity. Presentation of the data includes a poster as well as an oral presentation.

The abstract has been published online: View Source

Details on the poster presentation are as follows:

Abstract and Title: "Expitope 3.0 – An Advanced in silico Webtool Empowered with Machine Learning for Enhanced pHLA Epitope Prediction and Safety Assessment"

Authors: Sebastian Karg, Andrea Coluccio, Barbara Lösch, Dolores J Schendel, Dimitri Frishmann

Abstract Number: 98

Date/Time: Wednesday, May 3rd, 2023, 3:00 pm – 5.30 pm CET

Session: Postersession I

Details on the oral presentation are as follows:

Abstract and Title: "Expitope 3.0 – An Advanced in silico Webtool Empowered with Machine Learning for Enhanced pHLA Epitope Prediction and Safety Assessment"

Speaker: Dr. Barbara Lösch

Date/Time: Thursday, May 4th, 2023, 11.00 am – 11.15 am CET

Veracyte Announces Five Abstracts Providing Molecular Insights Into Prostate and Other Cancers To Be Presented at the 2023 ASCO Annual Meeting

On April 27, 2023 Veracyte, Inc. (Nasdaq: VCYT) reported that five abstracts providing new molecular insights into prostate and other cancers will be presented at the 2023 American Society of Clinical Oncology (ASCO) (Free ASCO Whitepaper) Annual Meeting, taking place in Chicago and online June 2-6 (Press release, Veracyte, APR 27, 2023, View Source [SID1234630628]). Three of the accepted abstracts leverage Veracyte’s Decipher GRID (Genomic Resource for Intelligent Discovery) database to explore potential opportunities for further personalizing treatment for patients with prostate cancer.

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"At Veracyte, we are committed to partnering with the scientific community to uncover new insights that may ultimately help further transform cancer care for patients," said Marc Stapley, Veracyte’s chief executive officer. "We particularly look forward to study findings being presented at ASCO (Free ASCO Whitepaper) that leverage our Decipher GRID database to explore differences in how patients with prostate cancer might respond to particular treatments based on their genomic profiles, and that demonstrate our deep scientific capabilities in immuno-oncology."

The following abstracts will be presented at the 2023 ASCO (Free ASCO Whitepaper) Annual Meeting:

Title: Longitudinal transcriptome profiling of localized hormone-sensitive tumors in treatment-naïve ENACT patients with prostate cancer with and without enzalutamide (ENZA)
Presenter: Ashley Ross, M.D., Ph.D., Northwestern University Feinberg School of Medicine
Abstract #: 5026
Format: Poster
Date/Time: June 3, 2023, 8:00-11:00 a.m. CT
Location: McCormick Place, Hall A (Poster #120)

Title: Basal-luminal subtyping of localized high-risk prostate cancer and benefit of adding docetaxel to definitive radiotherapy with androgen suppression in the NRG Oncology/RTOG 0521 phase III trial
Presenter: Ryan Phillips, M.D., Ph.D., Mayo Clinic
Abstract #: 5094
Format: Poster
Date/Time: June 3, 2023, 8:00-11:00 a.m. CT
Location: McCormick Place, Hall A (Poster #188)

Title: Transcriptomic heterogeneity of metastatic disease timing within metastatic castration-sensitive prostate cancer
First Author: Philip Sutera, M.D., Johns Hopkins University
Abstract #: e17083
Format: Publication Only

Title: Biology and performance of pre- and post-pembrolizumab (Pembro) vesical imaging–reporting and data system (VI-RADS) to predict the pathological response in muscle-invasive urothelial bladder cancer (MIBC): Full data analysis from a clinical trials pipeline
Presenter: Andrea Necchi, M.D., Vita-Salute San Raffaele University
Abstract #: 4591
Format: Poster
Date/Time: June 3, 2023, 8:00-11:00 a.m. CT
Location: McCormick Place, Hall A (Poster #83)

Title: FOLFOXIRI plus bevacizumab and atezolizumab as upfront treatment of unresectable metastatic colorectal cancer (mCRC): Updated and overall survival results of the phase II randomized AtezoTRIBE study.
Presenter: Carlotta Antoniotti, M.D., Ph.D., Department of Translational Research and New Technologies in Medicine and Surgery, University of Pisa & Unit of Medical Oncology 2, Azienda Ospedaliero-Universitaria Pisana
Abstract #: 3500
Format: Oral Presentation
Date/Time: June 4, 2023, 8:00 a.m. CT
Location: McCormick Place, Hall D2

Tempest to Report Early Results from Global Randomized Phase 1b/2 Combination Study of TPST-1120 in First-Line Hepatocellular Carcinoma

On April 27, 2023 Tempest Therapeutics, Inc. (Nasdaq: TPST), a clinical-stage oncology company developing first-in-class1 therapeutics that combine both targeted and immune-mediated mechanisms, reported that the company plans to report early data from its Phase 1b/2 combination study of TPST-1120 in first-line hepatocellular carcinoma in a premarket press release and webcast Friday, April 28, 2023 (Press release, Tempest Therapeutics, APR 27, 2023, View Source [SID1234630627]).

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Tempest will host a conference call accompanied by a slide presentation at 8:30 a.m. ET on Friday, April 28th. To join the conference call via phone and participate in the live Q&A session, please pre-register online here to receive a telephone number and unique passcode required to enter the call. The live webcast and audio archive of the presentation may be accessed on the investor section of the Tempest website at View Source The webcast will be available for replay for 30 days.

CHMP ISSUES POSITIVE OPINION FOR FUTIBATINIB FOR THE TREATMENT OF ADULTS WITH CHOLANGIOCARCINOMA

On April 27, 2023 Taiho Pharmaceutical Co., Ltd. and its European subsidiary Taiho Oncology Europe GmbH reported that the European Medicines Agency’s (EMA) Committee for Medicinal Products for Human Use (CHMP) has issued a positive opinion recommending the conditional marketing authorization (CMA) of futibatinib for the treatment of adult patients with locally advanced or metastatic cholangiocarcinoma(CCA) with a fibroblast growth factor receptor 2(FGFR2) fusion or rearrangement that have progressed after at least one prior line of systemic therapy (Press release, Taiho, APR 27, 2023, View Source [SID1234630624]).

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The CHMP’s opinion to recommend the use of futibatinib is now being reviewed by the full EMA. Final marketing authorizations for medical products in the European Union (EU) rests with the European Commission. Each year, approximately 6,000-8,000 individuals in Europe are diagnosed with CCA,1 a rare cancer of the bile ducts of the liver, and approximately 0.3-6 people per 100,000 individuals live with CCA worldwide.

"CCA is an aggressive cancer, and the current five-year survival rate is very poor, which underscores the need for new treatment options" said Peter Foertig, MD, Vice President, Medical Affairs, Taiho Oncology Europe. "We look forward to working with the European Medicines Agency as it reviews the application for marketing authorization."

The positive CHMP opinion on futibatinib is based on data from the pivotal Phase 2 FOENIX-CCA2 ※ trial in 103 patients with locally advanced or metastatic unresectable intrahepatic (inside the liver) CCA, harboring FGFR2 fusions or rearrangements who had received one or more prior lines of systemic therapy. Patients in the trial received futibatinib 20mg once daily until disease progression
or unacceptable toxicity. The trial’s primary endpoint was an objective response
rate (ORR).

※ FOENIX-CCA2:PHASE 1/2 STUDY OF TAS-120 IN PATIENTS WITH ADVANCED SOLID TUMORS Harboring FGF/FGFR Aberrations; FGFR Oral SElective Novel Inhibitor X [across] tumors

Results from the trial were published in the January 19, 2023, issue of The New England Journal of Medicine.

"As someone who treats patients with CCA, I am encouraged by these data and the positive news from CHMP," said Professor Arndt Vogel, MD, Senior Consultant, Department of Gastroenterology, Hepatology and Endocrinology, Hannover Medical School, Germany. "The study findings underscore the importance of molecular profiling for patients with CCA and other diseases whenever possible to potentially help improve outcomes. Indeed, the ESMO (Free ESMO Whitepaper) Clinical Practice Guidelines recommend FGFR inhibitors for the treatment of patients with CCA and FGFR2 fusions who have progressed after one or more prior lines of systemic therapy."

Takeshi Sagara Ph.D., Managing Director, Clinical Development and Medical Affairs, Discovery and Preclinical Research at Taiho Pharmaceutical, added "The global Taiho group will continue its efforts to bring futibatinib as a new treatment option to patients with CCA around the world, and the positive CHMP opinion represents a big step for Taiho in Europe to deliver innovative drugs to help patients with CCA in their journey".

About Futibatinib
Futibatinib (TAS-120) is an oral, potent, selective, and irreversible tyrosine kinase inhibitor of FGFR1, 2, 3 and 4 being studied as a potential treatment for patients with advanced solid tumors with FGFR1-4 genetic aberrations, including cholangiocarcinoma, who were previously treated with chemotherapy or other therapies. Futibatinib covalently binds to the ATP binding pocket of FGFR1-4
resulting in the inhibition of FGFR-mediated signal transduction pathways, reduced tumor cell proliferation in tumors with FGFR1-4 genetic aberrations.

In Japan, a new drug application for futibatinib has been submitted to the Japanese Ministry of Health, Labour and Welfare, as a treatment for previously treated locally advanced or metastatic biliary tract cancer harboring FGFR2 gene rearrangements, including gene fusions, on July 2022. Furthermore, in September 2022, the U.S. Food and Drug Administration (FDA) approved futibatinib for the treatment of adult patients with previously treated, unresectable, locally advanced or metastatic intrahepatic cholangiocarcinoma (iCCA) harboring fibroblast growth factor receptor 2 (FGFR2) gene fusions or other rearrangements.

Seagen Reports First Quarter 2023 Financial Results

On April 27, 2023 Seagen Inc. (Nasdaq:SGEN) (Seagen or the Company) reported financial results for the first quarter ended March 31, 2023 (Press release, Seagen, APR 27, 2023, View Source [SID1234630623]). The Company also highlighted performance across its approved product portfolio, development accomplishments, and progress across its differentiated oncology pipeline of innovative ADCs and targeted therapies.

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"Seagen delivered strong performance in the first quarter, with significant growth of 22 percent for both total revenue and net product sales, compared to 2022, driven by our multi-product commercial portfolio," said David Epstein, Chief Executive Officer of Seagen. "This month the FDA granted accelerated approval for PADCEV with KEYTRUDA for first-line treatment of patients with locally advanced or metastatic urothelial cancer who are ineligible for cisplatin. Additionally, the NCCN Guidelines for bladder cancer were recently updated to include the combination as a preferred regimen in this setting. This new indication substantially expands the number of addressable patients for this first-in-class therapy."

"In addition, this month we presented 17 abstracts at the American Association for Cancer Research (AACR) (Free AACR Whitepaper) Annual Meeting, including clinical and preclinical data from our early-stage pipeline," added Mr. Epstein. "At the upcoming American Society of Clinical Oncology (ASCO) (Free ASCO Whitepaper) Annual Meeting we will be presenting data from more than a dozen abstracts, including an oral presentation on long-term follow-up data from the combination of PADCEV and KEYTRUDA as well as updated data for SGN-B6A, a vedotin ADC targeting integrin beta-6, which is highly expressed in multiple solid tumors. We continue to link innovation to impact as we work to optimize the potential of our commercial products, prioritize the development of our most transformational pipeline assets and develop next-generation ADC technologies through the exploration of new payloads and linkers. Together with Pfizer, we will accelerate our ability to deliver transformative cancer medicines to more patients in need around the world."

PRODUCTS HIGHLIGHTS

PADCEV

Received FDA Accelerated Approval for PADCEV with KEYTRUDA for First-Line Treatment of Locally Advanced or Metastatic Urothelial Cancer (la/mUC): In April 2023, Seagen, Astellas and Merck announced the FDA granted PADCEV (enfortumab vedotin-ejfv) with KEYTRUDA (pembrolizumab) accelerated approval in the U.S. as a combination therapy for the treatment of adult patients with la/mUC who are not eligible to receive cisplatin-containing chemotherapy. It is the first treatment option combining an ADC with a PD-1 inhibitor in this patient population. Continued approval for this indication is contingent upon verification and description of clinical benefit in the EV-302 confirmatory trial, which has completed patient enrollment. An extension study has been initiated in China which continues to enroll patients.
NCCN Clinical Practice Guidelines in Oncology (NCCN Guidelines) for Bladder Cancer Updated to Include PADCEV and KEYTRUDA Combination as Preferred Regimen: In April 2023, based on the results of the EV-103 trial, the NCCN Guidelines were updated to include PADCEV with KEYTRUDA as a Preferred Regimen (Category 2A) for first-line therapy for patients with la/mUC who are not eligible to receive cisplatin-containing chemotherapy.
Biologics License Application (BLA) Accepted by China’s National Medical Products Administration (NMPA): In March 2023, the Center for Drug Evaluation (CDE) of the NMPA has accepted the BLA for PADCEV for the treatment of patients with la/mUC who received prior treatment with a PD-1/L1 inhibitor and platinum-based chemotherapy.
TUKYSA

Received FDA Accelerated Approval of TUKYSA in Combination with Trastuzumab for People with Previously Treated RAS Wild-Type, HER2-Positive Metastatic Colorectal Cancer: In January 2023, the FDAgranted accelerated approval to TUKYSA in combination with trastuzumab for adult patients with RAS wild-type, HER2-positive unresectable or metastatic colorectal cancer that has progressed following treatment with fluoropyrimidine-, oxaliplatin- and irinotecan-based chemotherapy. This is the first FDA-approved treatment specifically for HER2-positive metastatic colorectal cancer. Continued approval for this indication may be contingent upon verification and description of clinical benefit in confirmatory trials.
ADCETRIS

Received Orphan Drug Exclusivity (ODE) from FDA for Pediatric Indication: ODE provides seven years of market exclusivity for the recently approved indication of ADCETRIS for children with previously untreated high risk Hodgkin lymphoma. The FDA approved this new indication in November 2022.
TIVDAK

Completed Targeted Enrollment in Global Phase 3 Clinical Trial in Previously Treated Advanced Cervical Cancer: In February 2023, Seagen and our partner Genmab completed patient enrollment in the innovaTV 301 trial evaluating TIVDAK versus investigator’s choice of chemotherapy in previously treated recurrent or metastatic cervical cancer. The trial is intended to support global registrations and potentially serve as a confirmatory trial for the accelerated approval of TIVDAK in the U.S. An extension study has been initiated in China which continues to enroll patients.
Presented Data from innovaTV 207 Trial in Solid Tumors at the AACR (Free AACR Whitepaper) Annual Meeting: In April 2023, Seagen presented data from an interim analysis of Part C from the innovaTV 207 phase 2 study of TIVDAK given every 2 weeks in patients with recurrent or metastatic squamous cell carcinoma of the head and neck who have progressed on or after prior platinum combination, immunotherapy and targeted therapy, if eligible. Preliminary data based on the first 15 patients demonstrated encouraging antitumor activity with a confirmed overall response rate of 40% and a manageable safety profile.
PIPELINE PROGRAMS

Presented Multiple Abstracts on Early-Stage Pipeline at the AACR (Free AACR Whitepaper) Annual Meeting: Early-stage pipeline data included clinical, preclinical and discovery research programs. The first clinical data was presented for SEA-TGT that demonstrated a manageable and tolerable safety profile with initial monotherapy antitumor activity in solid tumors and lymphomas. In addition, data on multiple new ADC technologies were presented. These included the first preclinical data from Seagen and Sanofi for a novel topoisomerase I inhibitor ADC targeting CEACAM5, which demonstrated potent antitumor activity in patient-derived colorectal cancer models.

For additional information on Seagen’s pipeline, visit www.seagen.com/science/pipeline.
UPCOMING DATA PRESENTATIONS

Presenting Multiple Abstracts at the ASCO (Free ASCO Whitepaper) Annual Meeting: Seagen will present over a dozen abstracts at the ASCO (Free ASCO Whitepaper) Annual Meeting taking place June 2-6, demonstrating continued progress of the company’s clinical pipeline. Two oral presentations will highlight long-term follow-up data from a clinical trial of PADCEV in combination with KEYTRUDA, EV-103 dose-escalation and Cohort A, and initial data from a Phase 2 basket study of TUKYSA and trastuzumab in previously treated HER2-positive metastatic biliary tract cancer. Additionally, updated Phase 1 data will be presented for SGN-B6A.
CORPORATE HIGHLIGHT

Proposed Acquisition of Seagen by Pfizer: In March 2023, Seagen and Pfizer announced they have entered into a definitive merger agreement under which, on the terms and subject to the conditions thereof, Pfizer will acquire Seagen for $229 in cash per Seagen share for a total enterprise value of $43 billion. Pfizer and Seagen seek to accelerate the next generation of cancer breakthroughs and bring new solutions to patients by combining the power of Seagen’s ADC technology with the scale and strength of Pfizer’s capabilities and expertise. The Boards of Directors of both companies have unanimously approved the transaction. The companies expect to complete the transaction in late 2023 or early 2024, subject to fulfillment of customary closing conditions, including approval of Seagen’s stockholders and receipt of required regulatory approvals.
FIRST QUARTER AND THREE-MONTHS 2023 FINANCIAL RESULTS

Revenues: Total revenues for the first quarter of 2023 were $520 million, compared to $426 million for the same period in 2022, primarily driven by growth in net product sales.

Revenues included the following components:

Three months ended March 31,

(dollars in millions)

2023

2022

% Change

Total Net Product Sales

$

469

$

383

22

%

ADCETRIS

$

243

$

181

34

%

PADCEV

$

119

$

100

18

%

TUKYSA

$

87

$

90

(3

)%

TIVDAK

$

19

$

11

71

%

Royalty Revenues

$

30

$

28

7

%

Collaboration and License Agreement Revenues

$

21

$

15

38

%

Note: Sum of product sales may not equal total net product sales due to rounding. Percent change reflects actual (unrounded) values.

Net Product Sales: The increases in net product sales for the first quarter of 2023 compared to the same period in 2022 were driven by continued commercial execution. ADCETRIS performance was primarily attributed to volume growth, driven by greater use in frontline advanced Hodgkin lymphoma and an increase in diagnosis rates. PADCEV growth was primarily a result of additional eligible patients in the second-line, post-checkpoint maintenance setting for metastatic urothelial cancer, driven by continued penetration of checkpoint inhibitors in the first-line setting. TUKYSA performance reflects competitive dynamics in its breast cancer indication as well as early contributions from its colorectal cancer indication. TIVDAK growth reflects continued uptake in its current indication.
Royalty Revenues: Royalty revenues were primarily driven by sales of ADCETRIS outside the U.S. and Canada by Takeda as well as royalties from sales of Polivy (polatuzumab vedotin) by Roche, which is an ADC that uses Seagen technology.
Collaboration and License Agreement Revenues: The increase in collaboration and license agreement revenues was primarily driven by higher royalties from Astellas’ sales of PADCEV in its territory.
Cost of Sales: Cost of sales for the first quarter in 2023 were $112 million, compared to $88 million for the same period in 2022. The increases were primarily driven by higher sales of our medicines and the related gross profit share amounts owed to collaboration partners, which were $64 million in the first quarter in 2023, compared to $53 million for the same period in 2022. Cost of sales also reflects amortization of TUKYSA acquired in-process technology costs, third-party royalties owed for PADCEV and TUKYSA net product sales, and cost of products sold.

Research and Development (R&D) Expenses: R&D expenses for the first quarter in 2023 were $356 million, compared to $298 million for the same period in 2022 reflecting continued investment in clinical development of the Company’s approved drugs and pipeline programs.

Selling, General and Administrative (SG&A) Expenses: SG&A expenses for the first quarter in 2023 were $236 million, compared to $174 million for the same period in 2022. The increases in 2023 were driven by ongoing commercialization efforts, as well as $30 million in expenses associated with the pending acquisition by Pfizer and other corporate activities.

Non-cash, share-based compensation expense for the three months ended March 31, 2023 was $64 million, compared to $44 million for the same period in 2022.

Net Loss: Net loss for the first quarter of 2023 was $175 million, or $0.93 per diluted share. Net loss for the first quarter of 2022 was $136 million, or $0.74 per diluted share.

Cash and Investments: As of March 31, 2023, Seagen had $1.5 billion in cash and investments.

2023 FINANCIAL OUTLOOK AND CONFERENCE CALL

Given the pending acquisition of Seagen by Pfizer, Seagen will no longer be providing financial guidance for 2023 and will not be hosting its quarterly conference call and does not expect to do so for future quarters. Earnings materials are available publicly on the Investor Relations page of our website at investor.seagen.com. Please direct any questions to Seagen Investor Relations at the contact information below.