Vipergen Establishes DNA Encoded Library (DEL)-Based Drug Discovery Partnership with Theseus Pharmaceuticals Focused on Targeted Cancer Therapies

On April 4, 2022 Vipergen, a leading provider of small-molecule drug discovery services based on DNA-encoded library (DEL) technologies, reported the signing of a drug discovery agreement with Theseus Pharmaceuticals, a clinical-stage biopharmaceutical company focused on improving the lives of cancer patients through the discovery, development, and commercialization of transformative targeted therapies (Press release, Theseus Pharmaceuticals, APR 4, 2022, View Source [SID1234611425]). Under the terms of the agreement, Vipergen will apply its in-living-cell DNA-encoded library (DEL) screening platform to discover novel small-molecule compounds that bind to a selected Theseus kinase target. Theseus will select hits for potential development into targeted tyrosine kinase inhibitors (TKIs) and will retain exclusive rights to globally commercialize any products resulting from the collaboration. Financial details of the agreement were not disclosed.

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"Screening small-molecule libraries inside living cells—in a physiologically relevant context—is particularly important for success in developing cancer therapeutics," said Nils Hansen, PhD, Chief Executive Officer of Vipergen. "We are excited to apply our in-living-cell DEL screening technology to Theseus’ efforts to develop next-generation kinase inhibitors to transform the way cancer is treated."

Trishula Therapeutics Announces Oral Presentation on TTX-030 Anti-CD39 Antibody at American Association for Cancer Research (AACR) Annual Meeting

On April 4, 2022 Trishula Therapeutics, Inc., a clinical stage, privately held company developing TTX-030, a first-in-class anti-CD39 antibody in advanced cancers, reported preliminary results from an ongoing Phase 1 trial evaluating TTX-030 in combination with chemoimmunotherapy for the first-line treatment of patients with locally advanced or metastatic HER2- gastric or gastroesophageal junction (GEJ) cancer will be highlighted in an oral presentation at the American Association for Cancer Research (AACR) (Free AACR Whitepaper) Annual Meeting 2022 taking place in New Orleans, LA, April 8-13, 2022 (Press release, Trishula Therapeutics, APR 4, 2022, View Source [SID1234611424]).

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AACR Oral Presentation Details:

Title: Safety and efficacy of TTX-030, an anti-CD39 antibody, in combination with chemoimmunotherapy for the 1st line treatment of locally advanced or metastatic gastric/GEJ cancer.

Abstract Number: 8213

Session Title: Combination Immunotherapy Clinical Trials

Session Date and Time: Tuesday, April 12, 2022, 10:15 to 12:15 p.m., Central Time

Location: Hall B-C, Convention Center

Presentation Number: CT015

Vivace Therapeutics to Present New Data from Preclinical Combination Studies of VT3989 and Osimertinib at American Association for Cancer Research (AACR) Annual Meeting 2022

On April 4, 2022 Vivace Therapeutics, Inc., a small molecule discovery and development company developing first-in-class therapies targeting the Hippo pathway, reported that new preclinical data on the company’s transcriptional enhanced associate domain (TEAD) autopalmitoylation inhibitor, VT3989, will be presented at the American Association for Cancer Research (AACR) (Free AACR Whitepaper) Annual Meeting 2022 (Press release, Vivace Therapeurtics, APR 4, 2022, View Source [SID1234611423]). Presented findings will highlight results of research evaluating the combination of VT3989 and osimertinib (Tagrisso), an epidermal growth factor receptor (EGFR) inhibitor, in preclinical EGFR mutant tumor models. Study data demonstrated strong synergistic activity for the treatment combination as compared to osimertinib alone, as evidenced by enhanced efficacy and delayed tumor regrowth. The AACR (Free AACR Whitepaper) conference is being held April 8-13, 2022, in New Orleans, Louisiana.

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Vivace’s proprietary compounds inhibit palmitoylation of members of the TEAD protein family, including both covalent and non-covalent inhibitors. The company’s clinical candidate, VT3989, is currently in Phase 1 clinical trials. Pre-clinical research and development activities have demonstrated that the clinical candidate is active as a monotherapy against tumors that rely upon dysfunction of the Hippo pathway, and in combination with other anti-cancer therapies in additional tumor types.

Details of the company’s presentation at the AACR (Free AACR Whitepaper) conference are as follows:

Poster Presentation #5364:

Title: The TEAD autopalmitoylation inhibitor VT3989 improves efficacy and increases durability of efficacy of osimertinib in preclinical EGFR mutant tumor models
Presenting Author: Tracy Tang, Ph.D., vice president of biology, Vivace Therapeutics
Date/Time: Friday, April 8, 2022, 12:00 – 1:00 p.m. Central
Location: E-Poster Website

Accord BioPharma, in Partnership with Foresee Pharmaceuticals, Launches CAMCEVI™ (Leuprolide) Injection Emulsion in the U.S. for the Treatment of Advanced Prostate Cancer in Adults

On April 4, 2022 Accord BioPharma, the U.S. specialty division of Intas Pharmaceuticals, Ltd. focused on development of oncology, immunology, and critical care therapies, reported, in partnership with Foresee Pharmaceuticals Co., Ltd., the U.S. launch of CAMCEVI (leuprolide) 42mg injection emulsion for the treatment of advanced prostate cancer in adults (Press release, Foresee Pharmaceuticals, APR 4, 2022, View Source [SID1234611422]). The U.S. Food and Drug Administration approved the New Drug Application (NDA) of CAMCEVI from Foresee Pharmaceuticals on May 25, 2021. CAMCEVI 42 mg injection is exclusively licensed to Accord BioPharma in the U.S. for commercialization.

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"The U.S. launch of CAMCEVI validates the importance of Foresee’s pioneering Stabilized Injectable Formulation (SIF) technology and is a monumental step toward fulfilling our mission of improving on a standard of care," said Dr. Ben Chien, founder and Chairman of Foresee. "We know that Accord BioPharma shares in that important goal."

CAMCEVI is the first-ever ready-to-inject sterile formulation of leuprolide mesylate for subcutaneous injection that comes in a pre-filled syringe with no mixing required. In an open-label, single-arm study of 137 adults who received 42mg of CAMCEVI on Day 0 and Week 24, CAMCEVI offered consistent testosterone suppression to castrate levels after the initial injection, from Week 4 to Week 48.1 CAMCEVI should not be used in patients with hypersensitivity to GnRH or GnRH analogs due to possible anaphylactic reactions.1 The most common adverse reactions (≥10%) occurring during a median follow-up duration of 336 days were hot flush, hypertension, injection site reactions, upper respiratory tract infections, musculoskeletal pain, fatigue, and pain in extremity.1

"Accord Healthcare has been providing quality pharmaceutical products in the U.S. since the early 2000s. Through this partnership with Foresee on the launch of CAMCEVI, we are excited to formally launch Accord BioPharma with razor sharp focus on specialty pharmaceuticals, which will go beyond biology to bring more access to high-quality medicines to patients across the U.S.," said Binish Chudgar, Chairman, Accord Healthcare and Accord BioPharma.

"Foresee’s technology allows us to offer a therapy for advanced prostate cancer that is both effective and convenient for practitioners, with the pre-filled syringe providing simplified preparation that leads to an improved treatment experience for healthcare professionals," said Chrys Kokino, President of U.S. BioPharma at Accord BioPharma. "CAMCEVI marks an important example of our philosophy – going beyond biology – in action."

Important Safety Information: CAMCEVI, like other GnRH agonists, causes a transient increase in serum levels of testosterone during the first week of treatment which can cause transient worsening of symptoms. Patients with metastatic vertebral lesions and/or with urinary tract obstruction should be closely observed during the first few weeks of therapy. Hyperglycemia and an increased risk of developing diabetes have been reported in men receiving GnRH agonists. Blood glucose levels should be monitored and managed according to current clinical practice. Increased risk of myocardial infarction, sudden cardiac death, and stroke has been reported in association with the use of GnRH agonists. Patients should be monitored for cardiovascular disease and according to current clinical practice. Androgen deprivation therapy may prolong the QT interval. Convulsions have been reported in patients receiving GnRH agonists, like CAMCEVI. Monitor serum levels of testosterone following injection of CAMCEVI. Based on findings in animal studies and mechanism of action, CAMCEVI may cause fetal harm when administered to pregnant women. The most common (≥10%) adverse reactions during a median follow-up of 336 days were hot flush, hypertension, injection site reactions, upper respiratory tract infections, musculoskeletal pain, fatigue, and pain in extremities.

AI in Genomics Start-Up MNM Bioscience Gets nearly $1M Eureka Eurostars Funding for AI-Based Cancer Patient Stratification Tool

On April 4, 2022 MNM Bioscience, a technological start-up using genomic data and artificial intelligence algorithms to develop solutions for personalized medicine, reported that received an $800 000 grant from the Eureka’s Eurostars Programme (Press release, MNM Bioscience, APR 4, 2022, View Source [SID1234611421]). The program is a funding instrument dedicated for innovative SMEs, and will support the development of MNM’s unique patient stratification tool for ovarian cancer patients.

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This ambitious project will be realized in Consortium between MNM Bioscience and Macrogen Europe, a Dutch company focused on DNA sequencing and bioinformatics services.

The tool, named PARPiNDx (PARPindex), aims at better patient classification for the targeted anti-cancer therapy, increasing the chances to battle the disease through rapid implementation of the highly efficient drug. The tool selects patients who will respond to PARP inhibitors, a revolutionary drug family that is being successfully administered to patients with ovarian cancer, as well as several other cancer types, including pancreatic, breast and prostate cancers.

PARPiNDx is based on the genomic data derived from the whole genome sequencing data analyzed by AI-driven algorithms. PARPiNDx is not only selecting patients who will respond to PARPi, it is also identifying patients with intrinsic resistance to PARPi.

The consortium Agreement Was Signed 24th of March 2022.